SCHEMBL13628005

SCHEMBL13628005

O=C1/C(=N\O)c2cc(OC(F)(F)F)ccc2N1Cc1cccc([N+](=O)[O-])c1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 16/20 0.56
ALDH1A1 P00352 1/20 0.52
HPGD P15428 1/20 0.52
HTT P42858 1/20 0.52
CASP1 P29466 1/20 0.45
CASP3 P42574 1/20 0.45
CASP4 P49662 1/20 0.45
CASP7 P55210 1/20 0.45
CASP9 P55211 1/20 0.45
CASP6 P55212 1/20 0.45
CASP8 Q14790 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13910797 0.93 CHRM5 (0.56) CHRM5
SCHEMBL13627972 0.84 ALDH1A1 (0.57) ALDH1A1HPGDHTTCASP1CASP3
SCHEMBL13627951 0.82 ALDH1A1 (0.72) ALDH1A1HPGDHTTCASP1CASP3
SCHEMBL13628004 0.81 CHRM5 (0.74) CHRM5
SCHEMBL13627915 0.80 CASP1 (0.56) ALDH1A1HPGDHTTCASP1CASP3
SCHEMBL13628006 0.80 CHRM5 (0.63) CHRM5
SCHEMBL13627910 0.78 CASP1 (0.72) ALDH1A1HPGDHTTCASP1CASP3
SCHEMBL13627913 0.78 CASP1 (0.56) ALDH1A1HPGDHTTCASP1CASP3
SCHEMBL13627911 0.74 CASP3 (0.56) CHRM5ALDH1A1HPGDHTTCASP1
SCHEMBL13627887 0.73 MAPT (0.66) ALDH1A1HPGDHTTCASP1CASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612065-B2 Inhibitors of c-JUN N-terminal kinases (JNK) VERTEX PHARMACEUTICALS INCORPORATED (US) 2009-11-03 US disclosed
US-20080033022-A1 Inhibitors of c-Jun N-terminal kinases (JNK) SALITURO FRANCESCO G 2008-02-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080033022-A1 Inhibitors of c-Jun N-terminal kinases (JNK) MAP3K1, JUN, MAP3K7 CHRM5 4815/4885ALDH1A1 4310/4885HPGD 1551/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.