SCHEMBL13628709

SCHEMBL13628709

CCc1ccc(-c2ncn[nH]2)o1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.36
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
CHRM2 P08172 1/20 0.36
CHRM4 P08173 1/20 0.36
CHRM5 P08912 1/20 0.36
CHRM1 P11229 1/20 0.36
CHRM3 P20309 1/20 0.36
IDO1 P14902 6/20 0.35
ALDH1A1 P00352 2/20 0.34
ENPP2 Q13822 1/20 0.33
LMNA P02545 1/20 0.33
CYP1A2 P05177 1/20 0.31
CYP2E1 P05181 1/20 0.31
CYP2C8 P10632 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2A6 P11509 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2B6 P20813 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13628740 0.77 IDO1 (0.38) IDO1ALDH1A1ENPP2LMNA
SCHEMBL13628714 0.72 IDO1 (0.32) IDO1ENPP2PPARA
SCHEMBL13628700 0.72 ALOX5 (0.36) ALOX5PTGS1PTGS2CHRM2CHRM4
SCHEMBL10066946 0.66 METAP2 (0.44) IDO1ALDH1A1ENPP2LMNA
SCHEMBL13628742 0.66 CA12 (0.37) IDO1ALDH1A1ENPP2PPARA
SCHEMBL13628712 0.66 COMT (0.36) PTGS2IDO1ALDH1A1ENPP2CYP1A2
SCHEMBL13628718 0.66 ALOX5 (0.36) ALOX5PTGS1PTGS2CHRM2CHRM4
SCHEMBL45858 0.65
SCHEMBL3744556 0.65 IDO1 (0.50) IDO1ALDH1A1ENPP2PPARA
SCHEMBL15330895 0.64 CHRM2 (0.35) ALOX5PTGS1PTGS2CHRM2CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612070-B2 Heterocyclic compounds as antiinflammatory agents and cyclooxygenase inhibitors CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-11-03 US disclosed
US-7612070-B2 Heterocyclic compounds as antiinflammatory agents and cyclooxygenase inhibitors CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-11-03 US disclosed