SCHEMBL13628718

SCHEMBL13628718

CCc1ccc(-c2cnn[nH]2)o1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.36
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
CHRM2 P08172 1/20 0.36
CHRM4 P08173 1/20 0.36
CHRM5 P08912 1/20 0.36
CHRM1 P11229 1/20 0.36
CHRM3 P20309 1/20 0.36
CYP1A2 P05177 2/20 0.34
CYP2E1 P05181 2/20 0.34
CYP2C8 P10632 2/20 0.34
CYP2D6 P10635 2/20 0.34
CYP2A6 P11509 2/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2B6 P20813 2/20 0.34
CYP2C19 P33261 2/20 0.34
CYP3A4 P08684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13628747 0.77 MAPT (0.41) PTGS1PTGS2
SCHEMBL13628728 0.72 NOTUM (0.31)
SCHEMBL13628700 0.69 ALOX5 (0.36) ALOX5PTGS1PTGS2CHRM2CHRM4
SCHEMBL13628709 0.66 ALOX5 (0.36) ALOX5PTGS1PTGS2CHRM2CHRM4
SCHEMBL13628723 0.66 CYP2D6 (0.34) PTGS2CYP1A2CYP2E1CYP2C8CYP2D6
SCHEMBL45858 0.65
SCHEMBL805141 0.62 CYP2C19 (0.64) ALOX5PTGS1PTGS2CYP1A2CYP2E1
SCHEMBL13411815 0.61 POLB (0.33) CYP3A4
SCHEMBL13766598 0.61 TGFBR1 (0.33)
SCHEMBL10050008 0.61 ALDH1A1 (0.57) ALOX5PTGS1PTGS2CHRM2CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612070-B2 Heterocyclic compounds as antiinflammatory agents and cyclooxygenase inhibitors CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-11-03 US disclosed
US-7612070-B2 Heterocyclic compounds as antiinflammatory agents and cyclooxygenase inhibitors CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-11-03 US disclosed