SCHEMBL13628837

SCHEMBL13628837

COOSc1cnc2c(c1)cc(-c1ccco1)n2CC1CCCCC1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 7/20 0.39
ADORA1 P30542 7/20 0.39
ADORA3 P0DMS8 9/20 0.38
ADORA2B P29275 2/20 0.38
SCD5 Q86SK9 1/20 0.36
CCNA2 P20248 1/20 0.36
CDK2 P24941 1/20 0.36
CCNA1 P78396 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
CHRNB1 P11230 1/20 0.34
CHRNB2 P17787 1/20 0.34
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHRNB3 Q05901 1/20 0.34
PDE4B Q07343 2/20 0.33
MERTK Q12866 1/20 0.33
ALDH1A1 P00352 2/20 0.33
TP53 P04637 1/20 0.33
PDE7A Q13946 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13628828 0.83 ADORA3 (0.35) ADORA2AADORA1ADORA3ADORA2BSCD5
SCHEMBL13628827 0.83 NUAK1 (0.32) TDP1ALDH1A1
SCHEMBL2922408 0.79 ADORA2A (0.41) ADORA2AADORA1ADORA3ADORA2BSCD5
SCHEMBL13628834 0.78 ADORA3 (0.38) ADORA2AADORA1ADORA3ADORA2BTDP1
SCHEMBL13628819 0.78 CNR1 (0.43) ADORA2AADORA1ADORA3ADORA2BSCD5
SCHEMBL2925658 0.65 CNR2 (0.43) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL13628832 0.63 TRPC5 (0.38) TDP1ALDH1A1
SCHEMBL13628825 0.61 CYP1A2 (0.37) ALDH1A1TP53
SCHEMBL2927404 0.61 CNR2 (0.38) ALDH1A1
SCHEMBL7093005 0.59 SCD5 (0.55) ADORA2AADORA1ADORA3ADORA2BSCD5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612070-B2 Heterocyclic compounds as antiinflammatory agents and cyclooxygenase inhibitors CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-11-03 US disclosed