SCHEMBL13628834

SCHEMBL13628834

COOSc1cnc2c(c1)cc(-c1ccco1)n2Cc1ccccn1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 4/20 0.38
ADORA2A P29274 4/20 0.38
ADORA1 P30542 4/20 0.38
ADORA2B P29275 3/20 0.38
ALDH1A1 P00352 7/20 0.33
KDM4E B2RXH2 5/20 0.33
MAPT P10636 4/20 0.33
HPGD P15428 4/20 0.33
HSD17B10 Q99714 4/20 0.33
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
GAA P10253 2/20 0.33
CASP1 P29466 2/20 0.33
CASP7 P55210 2/20 0.33
TDP1 Q9NUW8 2/20 0.33
GLA P06280 1/20 0.33
GRIN1 Q05586 3/20 0.33
GRIN2B Q13224 3/20 0.33
POLB P06746 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13628819 0.83 CNR1 (0.43) ADORA3ADORA2AADORA1ADORA2BALDH1A1
SCHEMBL2928554 0.78 ADORA2A (0.39) ADORA3ADORA2AADORA1ADORA2BALDH1A1
SCHEMBL13628837 0.78 ADORA2A (0.39) ADORA3ADORA2AADORA1ADORA2BALDH1A1
SCHEMBL13628825 0.70 CYP1A2 (0.37) ALDH1A1MAPTHPGDHSD17B10SMN1; SMN2
SCHEMBL13628832 0.65 TRPC5 (0.38) ALDH1A1KDM4EMAPTHPGDHSD17B10
SCHEMBL13628865 0.63 RAB9A (0.35) ADORA2AGAA
SCHEMBL13628828 0.63 ADORA3 (0.35) ADORA3ADORA2AADORA1ADORA2BALDH1A1
SCHEMBL13628864 0.61 CYP1A2 (0.39) ALDH1A1HPGDHSD17B10SMN1; SMN2CASP1
SCHEMBL2928089 0.59 ALDH1A1 (0.51) ALDH1A1KDM4EMAPTHPGDHSD17B10
SCHEMBL30574744 0.57 KDM4E (0.49) ADORA3ADORA2AADORA1ADORA2BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612070-B2 Heterocyclic compounds as antiinflammatory agents and cyclooxygenase inhibitors CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-11-03 US disclosed