SCHEMBL13629592

SCHEMBL13629592

COc1ccc(-n2nccc2C(F)(F)F)cc1C=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.37
ALDH1A1 P00352 4/20 0.37
TSHR P16473 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
TUBB1 Q9H4B7 1/20 0.37
HPGD P15428 2/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
NPC1 O15118 1/20 0.35
POLB P06746 1/20 0.35
RAB9A P51151 1/20 0.35
FGFR1 P11362 1/20 0.35
LMNA P02545 2/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
PKM P14618 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
NTRK1 P04629 1/20 0.34
PTGS2 P35354 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13629598 0.81 PTGS2 (0.41) KDM4ECYP1A2CYP2C9LMNANTRK1
SCHEMBL310305 0.76 TACR1 (0.44) KDM4EALDH1A1HPGD
SCHEMBL3385723 0.73 PTGS2 (0.49) KDM4EALDH1A1TSHRCYP1A2CYP2C9
SCHEMBL27606848 0.72 ALDH1A1 (0.44) KDM4EALDH1A1TSHRTDP1HPGD
SCHEMBL7120569 0.70 MAPT (0.50) KDM4EALDH1A1TSHRTDP1HPGD
SCHEMBL1186123 0.70 ALDH1A1 (0.50) KDM4EALDH1A1TSHRTDP1TUBB1
SCHEMBL4205532 0.69 ATM (0.45) KDM4EALDH1A1TSHRTDP1HPGD
SCHEMBL7051253 0.69 ALDH1A1 (0.44) KDM4EALDH1A1TSHRTDP1TUBB1
SCHEMBL5193938 0.69 ALDH1A1 (0.42) KDM4EALDH1A1TSHRTDP1TUBB1
SCHEMBL8533478 0.69 LMNA (0.42) ALDH1A1TSHRHPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7622487-B2 Piperidine derivative, process for producing the same, and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-24 US disclosed
US-7622487-B2 Piperidine derivative, process for producing the same, and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-24 US disclosed