SCHEMBL13629598

SCHEMBL13629598

COc1ccc(-n2nccc2C(F)(F)F)cc1C

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.41
PTGS1 P23219 2/20 0.41
KDM4E B2RXH2 1/20 0.38
GAA P10253 1/20 0.37
CYP1A2 P05177 2/20 0.36
CYP2C9 P11712 2/20 0.36
GRM8 O00222 1/20 0.36
TACR1 P25103 1/20 0.36
GRM7 Q14831 1/20 0.36
NTRK1 P04629 1/20 0.36
ALOX15 P16050 1/20 0.35
UGCG Q16739 1/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
FUBP1 Q96AE4 1/20 0.34
NPBWR1 P48145 1/20 0.34
MCHR1 Q99705 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13629592 0.81 KDM4E (0.37) PTGS2KDM4ECYP1A2CYP2C9NTRK1
SCHEMBL16911136 0.80 ALOX15 (0.40) PTGS2PTGS1KDM4ECYP2C9ALOX15
SCHEMBL3385723 0.77 PTGS2 (0.49) PTGS2PTGS1KDM4ECYP1A2CYP2C9
SCHEMBL27606848 0.77 ALDH1A1 (0.44) KDM4ECYP1A2CYP2C9NTRK1LMNA
SCHEMBL28260479 0.75 KDM4E (0.47) PTGS2PTGS1KDM4ECYP2C9ALOX15
SCHEMBL16911833 0.73 UGCG (0.41) KDM4EGAAALOX15UGCGMAPT
SCHEMBL13629596 0.73 TACR1 (0.46) PTGS2PTGS1KDM4ETACR1MAPT
SCHEMBL4882670 0.72 KDM4E (0.42) PTGS2PTGS1KDM4ENTRK1
SCHEMBL2051437 0.72 NR3C2 (0.41) KDM4ECYP1A2CYP2C9UGCGMAPT
SCHEMBL16911329 0.71 RAB9A (0.40) KDM4EGAAALOX15LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7622487-B2 Piperidine derivative, process for producing the same, and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-24 US disclosed
US-7622487-B2 Piperidine derivative, process for producing the same, and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-24 US disclosed