SCHEMBL13635246

SCHEMBL13635246

COCCC(=O)Nc1ccc2[nH]nc(-c3cc4c(s3)C=CCC4)c2c1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ITK Q08881 7/20 0.44
AURKA O14965 4/20 0.42
AURKB Q96GD4 4/20 0.42
LRRK2 Q5S007 3/20 0.39
KDM4E B2RXH2 1/20 0.38
AAK1 Q2M2I8 1/20 0.38
MAPK10 P53779 1/20 0.37
TTK P33981 1/20 0.37
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2868617 0.78 MAPK10 (0.58) ITKAURKAAURKBLRRK2MAPK10
SCHEMBL13635414 0.77 MAPK10 (0.44) ITKMAPK10
SCHEMBL13635739 0.69 MAPK10 (0.38) ITKAURKAAURKBMAPK10TTK
SCHEMBL27539189 0.65 CLK2 (0.44) ITKAURKAAURKBLRRK2KDM4E
SCHEMBL2867353 0.65 ITK (0.60) ITKAURKAAURKBLRRK2TTK
SCHEMBL5383308 0.64 KMT2A (0.56) AURKAAURKBTTK
SCHEMBL2866702 0.63 MAPK10 (0.44) ITKKDM4EMAPK10
SCHEMBL5415164 0.63 ROCK2 (0.63)
SCHEMBL16025730 0.62 LRRK2 (0.55) LRRK2MAPK10
SCHEMBL2867196 0.62 MAPT (0.64) ITKAURKAAURKBLRRK2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1380576-B1 1H-INDAZOLE COMPOUNDS INHIBITING JNK EISAI R&D MAN CO LTD (JP) 2009-11-25 EP disclosed