SCHEMBL13637182

SCHEMBL13637182

COc1ccc2c(O)nc(-c3nc(C)co3)cc2c1C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 3/20 0.46
ESR1 P03372 3/20 0.34
ESR2 Q92731 3/20 0.34
KDM4E B2RXH2 4/20 0.33
ALDH1A1 P00352 4/20 0.33
RAD52 P43351 1/20 0.33
HPGD P15428 3/20 0.33
HSD17B10 Q99714 3/20 0.33
TSHR P16473 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
TDO2 P48775 1/20 0.32
MEN1 O00255 1/20 0.32
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 1/20 0.32
KMT2A Q03164 1/20 0.32
MCL1 Q07820 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13071901 0.85 PDE4B (0.34) PDE4BESR1ESR2KDM4EALDH1A1
SCHEMBL13637184 0.74 CYP3A4 (0.39) KDM4EALDH1A1HPGDHSD17B10TSHR
SCHEMBL7945510 0.68 MAPT (0.34) KDM4EALDH1A1HPGDL3MBTL1MEN1
SCHEMBL5592936 0.67 MAPK1 (0.55) PDE4BKDM4EALDH1A1HPGDHSD17B10
SCHEMBL14433126 0.62 PDE4B (0.41) PDE4BKDM4EALDH1A1HPGDHSD17B10
SCHEMBL8078744 0.62 ESR1 (0.49) ESR1ESR2MEN1KMT2A
SCHEMBL3624833 0.61 ENPP3 (0.43) PDE4BESR1ESR2KDM4EALDH1A1
SCHEMBL2237640 0.61 NQO2 (0.35) PDE4BESR1ESR2KDM4EALDH1A1
SCHEMBL15222168 0.61 IMPDH2 (0.51) PDE4BKDM4EALDH1A1RAD52HPGD
SCHEMBL2839768 0.60 ESR1 (0.38) PDE4BESR1ESR2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009142842-A2 NOVEL MACROCYCLIC INHIBITORS OF HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2009-11-26 WO disclosed