SCHEMBL13639002

SCHEMBL13639002

COCCNC(=O)c1cc(CCN2CCOCC2)ccc1NC(=O)c1csc(N2CC[C@H](OC)C2)n1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.42
ALDH1A1 P00352 2/20 0.42
MEN1 O00255 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
PDE5A O76074 2/20 0.39
GAA P10253 2/20 0.39
OPRK1 P41145 1/20 0.38
BCL3 P20749 1/20 0.38
WNT3A P56704 1/20 0.37
IRAK4 Q9NWZ3 1/20 0.37
LMNA P02545 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13634573 0.94 KMT2A (0.42) KMT2AALDH1A1MEN1CYP1A2CYP3A4
SCHEMBL13638912 0.93 KMT2A (0.47) KMT2AALDH1A1MEN1CYP1A2CYP3A4
SCHEMBL13634559 0.93 ALDH1A1 (0.41) KMT2AALDH1A1MEN1CYP1A2CYP3A4
SCHEMBL2770504 0.91 PIN1 (0.37) KMT2AMEN1OPRK1HRH3
SCHEMBL2774531 0.89 NAPEPLD (0.37) KMT2AMEN1HRH3
SCHEMBL2770287 0.89 PIN1 (0.36) KMT2AMEN1OPRK1HRH3
SCHEMBL15888680 0.89 PIN1 (0.36) KMT2AMEN1OPRK1HRH3
SCHEMBL13164108 0.89 KMT2A (0.38) KMT2AALDH1A1MEN1CYP1A2CYP3A4
SCHEMBL13639003 0.88 PIN1 (0.37) KMT2AMEN1OPRK1HRH3
SCHEMBL2772472 0.88 KMT2A (0.49) KMT2AALDH1A1MEN1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8304547-B2 Azolecarboxamide compound or salt thereof ASTELLAS PHARMA INC. (JP) 2012-11-06 US disclosed