SCHEMBL13639295

SCHEMBL13639295

COc1cc(Cl)ccc1-c1ccc2c(c1COc1cc(F)ccc1C)NC(=O)C(C)(C)N2

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IL6 P05231 8/20 0.53
PTGDR2 Q9Y5Y4 1/20 0.34
GRM5 P41594 1/20 0.34
FFAR1 O14842 1/20 0.33
FFAR4 Q5NUL3 1/20 0.33
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
MOGAT2 Q3SYC2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
KMT2A Q03164 1/20 0.32
GPBAR1 Q8TDU6 1/20 0.31
SCN9A Q15858 1/20 0.31
HTR2C P28335 2/20 0.31
TP53 P04637 1/20 0.31
MDM2 Q00987 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13639320 0.90 IL6 (0.63) IL6FFAR1FFAR4GRIN1GRIN2B
SCHEMBL13639301 0.85 IL6 (0.60) IL6FFAR1FFAR4GRIN1GRIN2B
SCHEMBL13639328 0.83 IL6 (0.55) IL6FFAR1FFAR4GPBAR1MDM2
SCHEMBL4580821 0.83 IL6 (0.76) IL6PTGDR2GRM5FFAR1FFAR4
SCHEMBL13639316 0.83 IL6 (0.57) IL6PTGDR2GRM5GRIN1GRIN2B
SCHEMBL4129581 0.83 IL6 (0.76) IL6PTGDR2GRM5FFAR1FFAR4
SCHEMBL4582029 0.83 IL6 (0.56) IL6KMT2A
SCHEMBL4145214 0.82 IL6 (0.46) IL6GRM5GRIN1GRIN2BMAPT
SCHEMBL13639334 0.82 IL6 (0.54) IL6ALDH1A1MAPTKMT2ATP53
SCHEMBL4142020 0.82 IL6 (0.42) IL6GRIN1GRIN2BMOGAT2MDM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1995242-B1 NOVEL 1,2,3,4-TETRAHYDROQUINOXALINE DERIVATIVE HAVING GLUCOCORTICOID RECEPTOR BINDING ACTIVITY SANTEN PHARMACEUTICAL CO LTD (JP) 2012-11-07 EP disclosed