SCHEMBL13639629

SCHEMBL13639629

COc1cc(Cl)ccc1/C(N)=C/c1cccc(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 1/20 0.44
RELA Q04206 1/20 0.43
ALDH1A1 P00352 3/20 0.40
GRIN2D O15399 2/20 0.40
GRIN3B O60391 2/20 0.40
GRIN1 Q05586 2/20 0.40
GRIN2A Q12879 2/20 0.40
GRIN2B Q13224 2/20 0.40
GRIN2C Q14957 2/20 0.40
GRIN3A Q8TCU5 2/20 0.40
KMT2A Q03164 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
TSHR P16473 1/20 0.39
XDH P47989 2/20 0.39
FLT1 P17948 1/20 0.39
FLT4 P35916 1/20 0.39
KDR P35968 1/20 0.39
FBP1 P09467 1/20 0.39
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12446116 0.81 GRIN1 (0.43) ALDH1A1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL2151674 0.80 KIF20A (0.54) ALDH1A1KMT2ANPC1RAB9AKDM4E
SCHEMBL2151685 0.80 KIF20A (0.54) ALDH1A1KMT2ANPC1RAB9AKDM4E
SCHEMBL5406529 0.75 NFE2L2 (0.57) NFE2L2RELAALDH1A1KMT2ANPC1
SCHEMBL6867023 0.73 GRIN2B (0.47) ALDH1A1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL12446542 0.72 MAOB (0.42) NFE2L2GRIN2BNPC1RAB9AFBP1
SCHEMBL1425701 0.72 FLT1 (0.54) ALDH1A1KMT2AFLT1FLT4KDR
SCHEMBL3436243 0.72 ALDH1A1 (0.66) ALDH1A1KMT2AFLT1FLT4KDR
SCHEMBL8118305 0.71 KIF20A (0.54) ALDH1A1KMT2AKDM4EMAPTMEN1
SCHEMBL13639623 0.70 KDM4E (0.52) KMT2ANPC1RAB9AFLT1FLT4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2340021-B1 SUBSTITUTED PYRROLIDINE-2-CARBOXAMIDES HOFFMANN LA ROCHE (CH) 2012-11-07 EP disclosed