SCHEMBL13639623

SCHEMBL13639623

COc1ccc(Cl)cc1/C=C(\N)c1ccc(Cl)cc1F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.52
CXCL12 P48061 1/20 0.44
SLC6A4 P31645 1/20 0.40
HTR3E A5X5Y0 1/20 0.39
HTR3B O95264 1/20 0.39
HTR3A P46098 1/20 0.39
HTR3D Q70Z44 1/20 0.39
HTR3C Q8WXA8 1/20 0.39
KMT2A Q03164 4/20 0.38
MAPT P10636 2/20 0.38
LMNA P02545 2/20 0.38
GAA P10253 1/20 0.38
CSF1R P07333 1/20 0.37
NUDT1 P36639 1/20 0.37
ERN1 O75460 1/20 0.37
MEN1 O00255 2/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
ATM Q13315 1/20 0.37
CYP11B1 P15538 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13639667 0.84 CYP11B2 (0.36) KDM4ECXCL12SLC6A4KMT2AMAPT
SCHEMBL2151666 0.80 KDM4E (0.55) KDM4ECXCL12KMT2AMAPTLMNA
SCHEMBL2151655 0.80 KDM4E (0.55) KDM4ECXCL12KMT2AMAPTLMNA
SCHEMBL12446099 0.74 ERN1 (0.37) CXCL12SLC6A4KMT2ALMNAERN1
SCHEMBL13639590 0.71 CYP11B2 (0.32) SLC6A4ERN1CYP11B1CYP11B2
SCHEMBL1765256 0.71 LMNA (0.50) SLC6A4HTR3EHTR3BHTR3AHTR3D
SCHEMBL12446116 0.71 GRIN1 (0.43) KDM4EKMT2AMAPTLMNAGAA
SCHEMBL13639648 0.71 TRPA1 (0.43) KDM4ECXCL12SLC6A4KMT2AMAPT
SCHEMBL13639629 0.70 NFE2L2 (0.44) KDM4EKMT2AMAPTGAAMEN1
SCHEMBL16953295 0.70 KDM4E (0.51) KDM4EHTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2340021-B1 SUBSTITUTED PYRROLIDINE-2-CARBOXAMIDES HOFFMANN LA ROCHE (CH) 2012-11-07 EP disclosed