SCHEMBL1364339

SCHEMBL1364339

Cc1c(C(=O)NCc2cccc(F)c2C2CC2)c2cccc(F)c2c(=O)n1Cc1ncco1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 8/20 0.41
SCD O00767 2/20 0.35
ALDH1A1 P00352 3/20 0.35
POLB P06746 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
SCN9A Q15858 2/20 0.33
RXFP1 Q9HBX9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1364957 0.88 S1PR3 (0.41) S1PR3SCDSCN9A
SCHEMBL1366992 0.86 ALDH1A1 (0.38) ALDH1A1POLBMAPTRXFP1
SCHEMBL1367487 0.84 ALDH1A1 (0.36) S1PR3ALDH1A1POLBLMNAMAPT
SCHEMBL2309159 0.83 S1PR3 (0.38) S1PR3
SCHEMBL1366943 0.82 ALDH1A1 (0.37) ALDH1A1POLBLMNAMAPTTSHR
SCHEMBL1367091 0.82 S1PR3 (0.43) S1PR3
SCHEMBL1364898 0.81 ALDH1A1 (0.35) S1PR3ALDH1A1POLBMAPT
SCHEMBL1367105 0.81 CYP1B1 (0.39) S1PR3SCN9A
SCHEMBL1945423 0.80 POLB (0.38) ALDH1A1POLBLMNAMAPTHPGD
SCHEMBL1943743 0.80 POLB (0.35) ALDH1A1POLBLMNAHPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110288120-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2011-11-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110288120-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS KCNK3, KCNQ3, KCNN3 S1PR3 559/4885SCD 4617/4885ALDH1A1 2697/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.