SCHEMBL1364898

SCHEMBL1364898

Cc1c(C(=O)NCc2cccc(F)c2C2CCC2)c2cccc(F)c2c(=O)n1Cc1ccoc1

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
S1PR3 Q99500 2/20 0.34
OPRK1 P41145 1/20 0.34
MAPT P10636 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
POLB P06746 1/20 0.33
APLNR P35414 1/20 0.32
CNR1 P21554 1/20 0.32
CNR2 P34972 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1367487 0.97 ALDH1A1 (0.36) ALDH1A1S1PR3MAPTL3MBTL1POLB
SCHEMBL1366992 0.84 ALDH1A1 (0.38) ALDH1A1MAPTL3MBTL1POLBAPLNR
SCHEMBL1367091 0.84 S1PR3 (0.43) S1PR3
SCHEMBL1364339 0.81 S1PR3 (0.41) ALDH1A1S1PR3MAPTPOLB
SCHEMBL1366943 0.81 ALDH1A1 (0.37) ALDH1A1MAPTL3MBTL1POLB
SCHEMBL2313628 0.79 HTR2A (0.36) ALDH1A1L3MBTL1POLB
SCHEMBL1366513 0.77 CYP2C9 (0.43) CNR1CNR2
SCHEMBL1945423 0.75 POLB (0.38) ALDH1A1MAPTPOLBAPLNR
SCHEMBL1366687 0.75 CYP2C9 (0.46)
SCHEMBL1943284 0.74 POLB (0.38) ALDH1A1MAPTPOLBAPLNR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110288120-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2011-11-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110288120-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS KCNK3, KCNQ3, KCNN3 ALDH1A1 2697/4885S1PR3 559/4885OPRK1 174/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.