SCHEMBL1367415

SCHEMBL1367415

CCc1nc2ccc(Cl)cc2c(Cl)c1C(=O)O

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FABP4 P15090 5/20 0.70
FABP3 P05413 4/20 0.70
FABP5 Q01469 4/20 0.70
ALDH1A1 P00352 3/20 0.49
CYP2C9 P11712 2/20 0.49
GAA P10253 1/20 0.49
MEN1 O00255 1/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
KMT2A Q03164 1/20 0.48
DHODH Q02127 8/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
POLB P06746 1/20 0.47
RECQL P46063 1/20 0.47
CASP6 P55212 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
PTGES O14684 1/20 0.43
ALOX5 P09917 1/20 0.43
HPGD P15428 1/20 0.43
CASP7 P55210 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11545050 0.93 FABP4 (0.64) FABP4FABP3FABP5ALDH1A1CYP2C9
SCHEMBL18285444 0.87 FABP4 (0.68) FABP4FABP3FABP5ALDH1A1CYP2C9
SCHEMBL10322427 0.86 RXFP1 (0.55) FABP4FABP3FABP5ALDH1A1CYP2C9
SCHEMBL6293298 0.85 FABP3 (0.61) FABP4FABP3FABP5ALDH1A1GAA
SCHEMBL18285435 0.82 FABP3 (0.52) FABP4FABP3FABP5ALDH1A1CYP2C9
SCHEMBL18285402 0.80 FABP3 (0.50) FABP4FABP3FABP5ALDH1A1GAA
SCHEMBL27638732 0.80 POLB (0.56) FABP4FABP3FABP5ALDH1A1CYP2C9
SCHEMBL537930 0.79 FABP4 (0.46) FABP4FABP3FABP5ALDH1A1CYP2C9
SCHEMBL3807965 0.77 FABP3 (0.47) FABP4FABP3FABP5ALDH1A1CYP2C9
SCHEMBL9869545 0.77 FABP4 (0.49) FABP4FABP3FABP5ALDH1A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11427582-B2 Ligands selective to alpha 6 subunit-containing GABAA receptors and their methods of use UWM RESEARCH FOUNDATION, INC. (US) 2022-08-30 US disclosed
US-20210047322-A1 LIGANDS SELECTIVE TO ALPHA 6 SUBUNIT-CONTAINING GABAA RECEPTORS AND THEIR METHODS OF USE NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2021-02-18 US disclosed
US-10865203-B2 Ligands selective to alpha 6 subunit-containing GABAA receptors and their methods of use UWM RESEARCH FOUNDATION, INC. (US) 2020-12-15 US disclosed
EP-3325479-B1 LIGANDS SELECTIVE TO ALPHA 6 SUBUNIT-CONTAINING GABAA RECEPTORS AND THEIR METHODS OF USE UWM RES FOUNDATION INC (US) 2020-12-02 EP disclosed
EP-3325479-A1 LIGANDS SELECTIVE TO ALPHA 6 SUBUNIT-CONTAINING GABAa RECEPTORS ANS THEIR METHODS OF USE UWM Research Foundation, Inc. (US) 2018-05-30 EP disclosed
US-20180134698-A1 LIGANDS SELECTIVE TO ALPHA 6 SUBUNIT-CONTAINING GABAA RECEPTORS AND THEIR METHODS OF USE NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2018-05-17 US disclosed
WO-2016196961-A1 LIGANDS SELECTIVE TO ALPHA 6 SUBUNIT-CONTAINING GABAA RECEPTORS ANS THEIR METHODS OF USE UWM RESEARCH FOUNDATION, INC. (US) 2016-12-08 WO disclosed
US-8889706-B2 Soluble mTOR complexes and modulators thereof WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2014-11-18 US disclosed
EP-2350053-B1 Modulators of MTOR Complexes WHITEHEAD BIOMEDICAL INST (US) 2013-12-11 EP disclosed
US-20130072485-A1 SOLUBLE MTOR COMPLEXES AND MODULATORS THEREOF DANA-FARBER CANCER INSTITUTE, INC. (US) 2013-03-21 US disclosed
US-8394818-B2 Soluble mTOR complexes and modulators thereof DANA-FARBER CANCER INSTITUTE, INC. (US) 2013-03-12 US disclosed
US-20110288091-A1 SOLUBLE MTOR COMPLEXES AND MODULATORS THEREOF WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2011-11-24 US disclosed
EP-2350053-A2 SOLUBLE MTOR COMPLEXES AND MODULATORS THEREOF Whitehead Institute For Biomedical Research (US) 2011-08-03 EP disclosed
WO-2010044885-A2 SOLUBLE MTOR COMPLEXES AND MODULATORS THEREOF WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2010-04-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210047322-A1 LIGANDS SELECTIVE TO ALPHA 6 SUBUNIT-CONTAINING GABAA RECEPTORS AND THEIR METHODS OF USE GABRA6, HTR6, GABRD FABP4 1209/4885FABP3 537/4885FABP5 611/4885
US-20130072485-A1 SOLUBLE MTOR COMPLEXES AND MODULATORS THEREOF MTOR, RICTOR, RPTOR FABP4 2231/4885FABP3 2903/4885FABP5 2100/4885
US-20180134698-A1 LIGANDS SELECTIVE TO ALPHA 6 SUBUNIT-CONTAINING GABAA RECEPTORS AND THEIR METHODS OF USE GABRA6, HTR6, GABRD FABP4 924/4885FABP3 427/4885FABP5 495/4885
US-11427582-B2 Ligands selective to alpha 6 subunit-containing GABAA receptors and their methods of use GABRA6, HTR6, GABRD FABP4 1209/4885FABP3 537/4885FABP5 611/4885
US-10865203-B2 Ligands selective to alpha 6 subunit-containing GABAA receptors and their methods of use GABRA6, HTR6, GABRD FABP4 924/4885FABP3 427/4885FABP5 495/4885
US-20110288091-A1 SOLUBLE MTOR COMPLEXES AND MODULATORS THEREOF MTOR, RICTOR, RPTOR FABP4 2231/4885FABP3 2903/4885FABP5 2100/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.