SCHEMBL13680450

SCHEMBL13680450

Cc1cccc(-c2ccc3[nH]c(=O)ccc3c2)n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.53
CA9 Q16790 2/20 0.53
F11 P03951 1/20 0.45
TGFBR1 P36897 2/20 0.45
CCR1 P32246 1/20 0.43
CCR8 P51685 1/20 0.43
CYP2A6 P11509 1/20 0.43
CA1 P00915 1/20 0.42
CA3 P07451 1/20 0.42
CA4 P22748 1/20 0.42
CA6 P23280 1/20 0.42
CA5A P35218 1/20 0.42
CA7 P43166 1/20 0.42
CA13 Q8N1Q1 1/20 0.42
CA14 Q9ULX7 1/20 0.42
CA5B Q9Y2D0 1/20 0.42
THRB P10828 1/20 0.41
MAPK1 P28482 2/20 0.40
SIK2 Q9H0K1 1/20 0.40
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680558 0.80 GRIA1 (0.59) TGFBR1CCR1CCR8CYP2A6SIK2
SCHEMBL13680569 0.78 NPC1 (0.54) CA12CA9TGFBR1CCR1CCR8
SCHEMBL4282655 0.78 CA12 (0.47) CA12CA9F11CYP2A6CA1
SCHEMBL13680545 0.77 CA12 (0.67) CA12CA9F11CA1CA3
SCHEMBL13680690 0.76 CCR1 (0.50) TGFBR1CCR1CCR8CYP2A6THRB
SCHEMBL15345000 0.75 CA12 (0.59) CA12CA9F11CCR1CCR8
SCHEMBL17505162 0.75 CA12 (0.51) CA12CA9F11CA1CA3
SCHEMBL13680856 0.75 CA12 (0.38) CA12CA9F11CA1CA3
SCHEMBL16573987 0.74 CA12 (0.73) CA12CA9F11CA1CA3
Hydrochloric Acid SCHEMBL11122791 0.74 MAPT (0.47) CA12CA9F11THRBHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed