SCHEMBL13680856

SCHEMBL13680856

O=CCCc1cccc(-c2ccc3[nH]c(=O)ccc3c2)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.38
CA9 Q16790 2/20 0.38
F11 P03951 1/20 0.38
CA1 P00915 1/20 0.36
CA3 P07451 1/20 0.36
CA4 P22748 1/20 0.36
CA6 P23280 1/20 0.36
CA5A P35218 1/20 0.36
CA7 P43166 1/20 0.36
CA13 Q8N1Q1 1/20 0.36
CA14 Q9ULX7 1/20 0.36
CA5B Q9Y2D0 1/20 0.36
HPGD P15428 1/20 0.35
AR P10275 1/20 0.35
POLB P06746 2/20 0.34
PKM P14618 1/20 0.34
PDE3B Q13370 2/20 0.33
PDE3A Q14432 2/20 0.33
TBXAS1 P24557 1/20 0.33
PIK3CD O00329 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13681003 0.77 HRH3 (0.39) CA12CA9F11CA1CA3
SCHEMBL13680450 0.75 CA12 (0.53) CA12CA9F11CA1CA3
SCHEMBL13680977 0.72 CA12 (0.40) CA12CA9F11CA1CA3
SCHEMBL3854280 0.72 MEN1 (0.50) PDE10A
SCHEMBL13680834 0.72 PDE10A (0.39) HPGDPOLBIRAK4PDE10A
SCHEMBL13680817 0.71 ALDH1A1 (0.47) HPGDMAPK1PDE10A
SCHEMBL4282655 0.71 CA12 (0.47) CA12CA9F11CA1CA3
SCHEMBL13680855 0.70 IRAK4 (0.42) ARIRAK4
SCHEMBL13680831 0.69 PDE10A (0.37) PDE10A
SCHEMBL13680846 0.69 MAPT (0.40) KDRPDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed