SCHEMBL13680569

SCHEMBL13680569

Cc1cccc(-c2ccc3[nH]ccc3c2)n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.54
TGFBR1 P36897 2/20 0.51
BRD4 O60885 1/20 0.50
FYN P06241 1/20 0.49
CCR1 P32246 1/20 0.48
CCR8 P51685 1/20 0.48
ADORA2A P29274 1/20 0.48
ADORA1 P30542 1/20 0.48
NISCH Q9Y2I1 1/20 0.45
CYP17A1 P05093 1/20 0.44
CYP11B1 P15538 1/20 0.44
CYP11B2 P19099 1/20 0.44
BPTF Q12830 1/20 0.44
CYP2A6 P11509 1/20 0.44
GUSB P08236 2/20 0.43
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.43
PARP10 Q53GL7 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680450 0.78 CA12 (0.53) TGFBR1CCR1CCR8CYP2A6CA12
SCHEMBL13680563 0.78 TGFBR1 (0.77) TGFBR1
SCHEMBL4873744 0.77 TGFBR1 (0.42) NPC1TGFBR1BRD4FYNADORA2A
SCHEMBL13680562 0.76 CDK8 (0.58) BRD4
SCHEMBL17149330 0.76 IMPDH2 (0.54) NPC1BRD4FYNADORA2AADORA1
SCHEMBL7330846 0.76 NPC1 (0.58) NPC1BRD4FYNADORA2AADORA1
SCHEMBL9231655 0.76 NPC1 (0.68) NPC1BRD4FYNADORA2AADORA1
SCHEMBL11990860 0.76 CCR1 (0.68) TGFBR1CCR1CCR8CYP2A6
SCHEMBL13680558 0.75 GRIA1 (0.59) TGFBR1CCR1CCR8CYP2A6
SCHEMBL5850255 0.75 NPC1 (0.79) NPC1BRD4FYNNISCHCYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed