SCHEMBL13680629

SCHEMBL13680629

Cc1csc(-c2ccc3c(c2)CNC3=O)n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.52
CLK4 Q9HAZ1 2/20 0.52
DAPK3 O43293 1/20 0.52
NTRK1 P04629 1/20 0.52
PIM1 P11309 1/20 0.52
FLT3 P36888 1/20 0.52
ROCK1 Q13464 1/20 0.52
BRAF P15056 1/20 0.47
PRF1 P14222 5/20 0.45
PRKCI P41743 1/20 0.44
TGFBR1 P36897 1/20 0.43
ACVR1 Q04771 1/20 0.43
TBK1 Q9UHD2 1/20 0.42
GABRA1 P14867 2/20 0.41
GABRG2 P18507 2/20 0.41
GABRB3 P28472 2/20 0.41
GABRA5 P31644 2/20 0.41
GABRA3 P34903 2/20 0.41
GABRA2 P47869 2/20 0.41
CYP2E1 P05181 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31267870 0.78 CLK4 (0.52) GSK3BCLK4DAPK3NTRK1PIM1
SCHEMBL13680735 0.78 HSD17B1 (0.48) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL13681013 0.78 PRF1 (0.43) GSK3BCLK4DAPK3NTRK1PIM1
SCHEMBL15984853 0.76 GSK3B (0.56) GSK3BCLK4DAPK3NTRK1PIM1
SCHEMBL13680620 0.76 PRF1 (0.55) PRF1GLA
SCHEMBL3873312 0.76 CYP2E1 (0.43) TGFBR1GABRA1GABRG2GABRB3GABRA5
SCHEMBL13680577 0.74 CLK4 (0.53) GSK3BCLK4DAPK3NTRK1PIM1
SCHEMBL20923873 0.73 PRF1 (0.62) GSK3BCLK4DAPK3NTRK1PIM1
SCHEMBL13680630 0.73 PDE3B (0.57) TGFBR1ACVR1
SCHEMBL13680628 0.71 CRBN (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed