SCHEMBL13680735

SCHEMBL13680735

Cc1csc(-c2ccc3c(c2)CCC3=O)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 4/20 0.48
CYP1A2 P05177 1/20 0.46
CYP11B1 P15538 1/20 0.46
CYP11B2 P19099 1/20 0.46
PTGS1 P23219 1/20 0.43
PTGS2 P35354 1/20 0.43
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
HSD17B10 Q99714 1/20 0.41
PGR P06401 1/20 0.41
GLA P06280 1/20 0.41
GABRA1 P14867 5/20 0.40
GABRG2 P18507 5/20 0.40
GABRB3 P28472 5/20 0.40
GABRA3 P34903 5/20 0.40
GABRA5 P31644 3/20 0.40
GABRA2 P47869 3/20 0.40
CYP2E1 P05181 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2A6 P11509 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680620 0.78 PRF1 (0.55) PTGS1PTGS2GLAMAPT
SCHEMBL13680629 0.78 GSK3B (0.52) GLAGABRA1GABRG2GABRB3GABRA3
SCHEMBL13681043 0.77 HSD17B1 (0.42) HSD17B1CYP1A2CYP11B1CYP11B2CASP1
SCHEMBL2439734 0.74 CYP1A2 (0.49) HSD17B1CYP1A2CYP11B1CYP11B2PTGS2
SCHEMBL28655414 0.74 HSD17B1 (0.78) HSD17B1CYP1A2CYP11B1CYP11B2CASP1
SCHEMBL2443326 0.74 CYP1A2 (0.51) HSD17B1CYP1A2CYP11B1CYP11B2PTGS1
SCHEMBL13680668 0.72 CYP1A2 (0.50) HSD17B1CYP1A2CYP11B1CYP11B2CASP1
SCHEMBL2432038 0.72 CYP1A2 (0.50) HSD17B1CYP1A2CYP11B1CYP11B2CASP1
SCHEMBL13680623 0.72 NPC1 (0.41) GLAGABRA1GABRG2GABRB3GABRA3
SCHEMBL13680630 0.72 PDE3B (0.57) CYP1A2CYP11B1CYP11B2PGRNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed