SCHEMBL13680650

SCHEMBL13680650

CSc1ncc(-c2cccc(C)c2)cn1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ENPP3 O14638 1/20 0.42
IDO1 P14902 1/20 0.42
METAP2 P50579 1/20 0.42
NR1I3 Q14994 1/20 0.42
RAB9A P51151 2/20 0.41
MAP4K4 O95819 2/20 0.41
ACHE P22303 2/20 0.40
MAPK14 Q16539 1/20 0.40
BCHE P06276 1/20 0.40
ADORA1 P30542 1/20 0.40
NPC1 O15118 1/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
ATM Q13315 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680651 0.80 IDO1 (0.47) ENPP3IDO1METAP2RAB9AMAP4K4
SCHEMBL6885681 0.78 RAB9A (0.54) RAB9ANPC1HPGDSMN1; SMN2ALDH1A1
SCHEMBL13040 0.77 MAP4K4 (0.66) IDO1METAP2RAB9AMAP4K4ADORA1
SCHEMBL15344198 0.77 EGLN1 (0.47) IDO1METAP2RAB9AMAP4K4ACHE
SCHEMBL13681263 0.76 MAP4K4 (0.43) ENPP3IDO1METAP2RAB9AMAP4K4
SCHEMBL13680652 0.76 RAB9A (0.63) IDO1METAP2RAB9AACHEBCHE
SCHEMBL29373699 0.74 ACHE (0.69) ENPP3IDO1METAP2RAB9AMAP4K4
SCHEMBL31471473 0.74 ACHE (0.69) ENPP3IDO1METAP2RAB9AMAP4K4
SCHEMBL301247 0.74 ACHE (0.69) ENPP3IDO1METAP2RAB9AMAP4K4
SCHEMBL13680543 0.74 FTO (0.50) IDO1METAP2RAB9AMAP4K4ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed