SCHEMBL13680668

SCHEMBL13680668

Cc1cccc(-c2ccc3c(c2)CCC3=O)n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.50
CYP11B1 P15538 1/20 0.50
CYP11B2 P19099 1/20 0.50
HSD17B1 P14061 4/20 0.49
CCR1 P32246 1/20 0.43
CCR8 P51685 1/20 0.43
GRM1 Q13255 1/20 0.43
CYP2A6 P11509 1/20 0.43
CASP1 P29466 1/20 0.42
CASP7 P55210 1/20 0.42
HSD17B10 Q99714 1/20 0.42
PGR P06401 1/20 0.42
PARP10 Q53GL7 2/20 0.42
PARP11 Q9NR21 2/20 0.42
TGFBR1 P36897 1/20 0.41
SIK2 Q9H0K1 2/20 0.40
GRM5 P41594 1/20 0.40
STK4 Q13043 1/20 0.39
STK3 Q13188 1/20 0.39
STK26 Q9P289 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680566 0.78 PRF1 (0.52)
SCHEMBL2448407 0.78 KDM4E (0.49) CYP1A2CYP11B1CYP11B2HSD17B1GRM1
SCHEMBL13680577 0.77 CLK4 (0.53) CYP2A6PARP10PARP11TGFBR1GRM5
SCHEMBL2432038 0.77 CYP1A2 (0.50) CYP1A2CYP11B1CYP11B2HSD17B1GRM1
SCHEMBL19734014 0.76 CYP1A2 (0.56) CYP1A2CYP11B1CYP11B2HSD17B1GRM1
SCHEMBL3630871 0.75 HSD17B1 (0.54) CYP1A2CYP11B1CYP11B2HSD17B1GRM1
SCHEMBL13680642 0.75 PARP10 (0.64) CYP1A2CYP11B1CYP11B2HSD17B1GRM1
SCHEMBL28655414 0.75 HSD17B1 (0.78) CYP1A2CYP11B1CYP11B2HSD17B1GRM1
SCHEMBL20865266 0.73 CCR1 (0.54) CCR1CCR8CYP2A6TGFBR1
SCHEMBL1747435 0.73 HSD17B1 (0.69) CYP1A2CYP11B1CYP11B2HSD17B1GRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed