SCHEMBL13680675

SCHEMBL13680675

CNc1ncc(-c2cccc(C)n2)cn1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.52
CCR8 P51685 1/20 0.52
CYP2A6 P11509 1/20 0.50
MAP4K4 O95819 1/20 0.47
SIK2 Q9H0K1 9/20 0.47
STK3 Q13188 8/20 0.46
STK26 Q9P289 8/20 0.46
STK24 Q9Y6E0 8/20 0.46
STK4 Q13043 7/20 0.46
MAPT P10636 1/20 0.43
METAP2 P50579 1/20 0.42
PAK1 Q13153 1/20 0.40
GRM5 P41594 2/20 0.40
TGFBR1 P36897 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680679 0.81 CCR1 (0.60) CCR1CCR8CYP2A6METAP2GRM5
SCHEMBL13680676 0.79 CYP2A6 (0.47) CCR1CCR8CYP2A6MAPTGRM5
SCHEMBL13680673 0.78 CCR1 (0.56) CCR1CCR8CYP2A6MAP4K4METAP2
SCHEMBL13680686 0.77 CYP2A6 (0.45) CCR1CCR8CYP2A6SIK2MAPT
SCHEMBL13680677 0.76 CCR1 (0.54) CCR1CCR8CYP2A6METAP2GRM5
SCHEMBL30146674 0.76 CYP2A6 (0.65) CCR1CCR8CYP2A6METAP2GRM5
SCHEMBL3421947 0.76 CYP2A6 (0.65) CCR1CCR8CYP2A6METAP2GRM5
SCHEMBL13680680 0.75 CYP2A6 (0.54) CCR1CCR8CYP2A6METAP2TGFBR1
SCHEMBL13680586 0.75 CCR1 (0.52) CCR1CCR8CYP2A6MAPTMETAP2
SCHEMBL13680674 0.75 CCR1 (0.52) CCR1CCR8CYP2A6METAP2GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed