SCHEMBL13680686

SCHEMBL13680686

COC(=O)Nc1ncc(-c2cccc(C)n2)cn1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.45
GRM5 P41594 2/20 0.45
CCR1 P32246 1/20 0.42
CCR8 P51685 1/20 0.42
RAB9A P51151 2/20 0.41
KMT2A Q03164 2/20 0.39
AAK1 Q2M2I8 2/20 0.39
MEN1 O00255 1/20 0.39
HTT P42858 1/20 0.39
EGFR P00533 1/20 0.39
BTK Q06187 1/20 0.39
MAPT P10636 2/20 0.38
ALOX5 P09917 1/20 0.38
TGFBR1 P36897 2/20 0.37
NPC1 O15118 1/20 0.37
GBA1 P04062 1/20 0.37
TSHR P16473 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
SIK2 Q9H0K1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680676 0.85 CYP2A6 (0.47) CYP2A6GRM5CCR1CCR8RAB9A
SCHEMBL13537053 0.79 SMN1; SMN2 (0.49) CYP2A6CCR1CCR8RAB9AKMT2A
SCHEMBL13680544 0.77 CNR1 (0.51) CYP2A6RAB9AKMT2AMEN1MAPT
SCHEMBL13680675 0.77 CCR1 (0.52) CYP2A6GRM5CCR1CCR8MAPT
SCHEMBL13680554 0.77 GRM5 (0.53) CYP2A6GRM5CCR1CCR8KMT2A
SCHEMBL13680657 0.75 FAAH (0.46) AAK1
SCHEMBL13680678 0.74 CYP2A6 (0.51) CYP2A6GRM5CCR1CCR8RAB9A
SCHEMBL13680586 0.73 CCR1 (0.52) CYP2A6GRM5CCR1CCR8KMT2A
SCHEMBL13680679 0.72 CCR1 (0.60) CYP2A6GRM5CCR1CCR8RAB9A
SCHEMBL8241210 0.72 HPGD (0.46) RAB9AKMT2AMEN1HTTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed