SCHEMBL13680748

SCHEMBL13680748

COC(=O)Nc1ncc(-c2nc(C)cs2)cn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2E1 P05181 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2A6 P11509 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2B6 P20813 1/20 0.40
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
KDM4E B2RXH2 2/20 0.38
GAA P10253 2/20 0.38
TGFBR1 P36897 1/20 0.38
MAPT P10636 1/20 0.37
TSHR P16473 1/20 0.37
HPGDS O60760 3/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
HSD17B10 Q99714 1/20 0.37
RCE1 Q9Y256 1/20 0.37
PIK3C3 Q8NEB9 1/20 0.36
POLB P06746 1/20 0.36
AOC3 Q16853 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680747 0.85 CYP2C9 (0.42) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL13681291 0.82 CYP2E1 (0.39) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL13680489 0.78 SMN1; SMN2 (0.47) NPC1RAB9AKDM4EGAAMAPT
SCHEMBL13681058 0.77 MAPT (0.37) KDM4EGAAMAPTALDH1A1HPGD
SCHEMBL13680746 0.77 CYP3A4 (0.47) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL13680742 0.74 CYP2E1 (0.45) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL13680615 0.73 CYP2E1 (0.47) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL13680540 0.73 DYRK1A (0.52) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL13680744 0.72 CYP3A4 (0.53) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL8241210 0.72 HPGD (0.46) CYP3A4RAB9AKDM4EMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed