SCHEMBL13680747

SCHEMBL13680747

CC(=O)Nc1ncc(-c2nc(C)cs2)cn1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.42
CYP2E1 P05181 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2A6 P11509 1/20 0.42
CYP2B6 P20813 1/20 0.42
TGFBR1 P36897 2/20 0.40
NPC1 O15118 4/20 0.40
RAB9A P51151 4/20 0.40
KDM4E B2RXH2 1/20 0.40
GAA P10253 1/20 0.40
TKT P29401 1/20 0.39
MAPT P10636 1/20 0.39
TSHR P16473 1/20 0.38
PIK3C3 Q8NEB9 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C19 P33261 1/20 0.38
HPGDS O60760 1/20 0.38
SLC12A5 Q9H2X9 1/20 0.37
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680748 0.85 CYP2E1 (0.40) CYP2C9CYP2E1CYP3A4CYP2A6CYP2B6
SCHEMBL13681291 0.84 CYP2E1 (0.39) CYP2C9CYP2E1CYP3A4CYP2A6CYP2B6
SCHEMBL13680742 0.80 CYP2E1 (0.45) CYP2C9CYP2E1CYP3A4CYP2A6CYP2B6
SCHEMBL13680746 0.79 CYP3A4 (0.47) CYP2C9CYP2E1CYP3A4CYP2A6CYP2B6
SCHEMBL13680522 0.77 RAB9A (0.55) NPC1RAB9AKDM4EGAAMAPT
SCHEMBL13681047 0.76 ADRB2 (0.40) RAB9AKDM4ETKTSREBF2
SCHEMBL13680744 0.75 CYP3A4 (0.53) CYP2C9CYP2E1CYP3A4CYP2A6CYP2B6
SCHEMBL30585336 0.72 TGFBR1 (0.45) TGFBR1NPC1RAB9AKDM4EGAA
SCHEMBL13680738 0.72 CYP3A4 (0.50) CYP2C9CYP2E1CYP3A4CYP2A6CYP2B6
SCHEMBL13304496 0.70 ADORA3 (0.46) CYP2C9RAB9AKDM4EMAPTPIK3C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed