SCHEMBL13680822

SCHEMBL13680822

COc1ccc(CCC=O)nc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.38
ALDH1A1 P00352 1/20 0.37
CYP2A6 P11509 1/20 0.37
MCHR1 Q99705 2/20 0.36
MBOAT4 Q96T53 1/20 0.36
TUBB4A P04350 1/20 0.36
TUBB P07437 1/20 0.36
TUBA3C P0DPH7 1/20 0.36
TUBA1B P68363 1/20 0.36
TUBA4A P68366 1/20 0.36
TUBB4B P68371 1/20 0.36
TUBB3 Q13509 1/20 0.36
TUBB2A Q13885 1/20 0.36
TUBB8 Q3ZCM7 1/20 0.36
TUBA3E Q6PEY2 1/20 0.36
TUBA1A Q71U36 1/20 0.36
TUBA1C Q9BQE3 1/20 0.36
TUBB6 Q9BUF5 1/20 0.36
TUBB2B Q9BVA1 1/20 0.36
TUBB1 Q9H4B7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3362831 0.82 ALDH1A1 (0.39) CYP3A4ALDH1A1CYP2A6MBOAT4TUBB4A
SCHEMBL18851549 0.78 MCHR1 (0.43) CYP3A4ALDH1A1MCHR1MBOAT4MAPT
SCHEMBL24928598 0.78 ADORA2A (0.41) CYP3A4ALDH1A1CYP2A6MBOAT4TUBB4A
SCHEMBL6197859 0.77 CCR1 (0.40) CYP3A4ALDH1A1CYP2A6MAPTADORA2A
SCHEMBL31338938 0.77 MCHR1 (0.42) CYP3A4MCHR1MBOAT4TUBB4ATUBB
SCHEMBL25253178 0.77 PTGS2 (0.40) CYP3A4MCHR1MBOAT4ADORA2ANPC1
SCHEMBL1025383 0.77 TAAR1 (0.52) CYP3A4ALDH1A1MCHR1MBOAT4MAPT
SCHEMBL28114840 0.76 NAAA (0.40) ALDH1A1CYP2A6MCHR1MBOAT4TUBB4A
SCHEMBL17541075 0.76 CA12 (0.40) CYP3A4ALDH1A1MBOAT4TUBB4ATUBB
SCHEMBL26807141 0.75 ACACB (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed