SCHEMBL13684451

SCHEMBL13684451

CC(C)NC(=O)NC(CN1CCCS1(=O)=O)C(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PER2 O15055 16/20 0.40
CRY1 Q16526 16/20 0.40
CRY2 Q49AN0 16/20 0.40
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
KMT2A Q03164 1/20 0.33
SIGMAR1 Q99720 1/20 0.32
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13127922 0.90 PER2 (0.37) PER2CRY1CRY2
SCHEMBL13792023 0.84 PER2 (0.41) PER2CRY1CRY2
SCHEMBL13622636 0.81 CTSK (0.39) PER2CRY1CRY2
SCHEMBL8282004 0.81 CTSK (0.39) PER2CRY1CRY2
SCHEMBL13791794 0.80 CRY1 (0.38) PER2CRY1CRY2
SCHEMBL8270963 0.78 PER2 (0.41) PER2CRY1CRY2
SCHEMBL13633039 0.78 PER2 (0.44) PER2CRY1CRY2
SCHEMBL13622674 0.77 CTSK (0.41) PER2CRY1CRY2
SCHEMBL8282033 0.77 CTSK (0.41) PER2CRY1CRY2
SCHEMBL8279628 0.75 CRY1 (0.39) PER2CRY1CRY2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7592419-B2 Macrocyclic inhibitors of hepatitis C virus NS3-serine protease SCHERING CORPORATION (US) 2009-09-22 US disclosed