SCHEMBL13685302

SCHEMBL13685302

CC(C)(C)ON(C=O)Cc1ccc(B(O)O)cc1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LPL P06858 7/20 0.41
LIPG Q9Y5X9 7/20 0.41
KDM4E B2RXH2 1/20 0.37
CA2 P00918 3/20 0.37
CA1 P00915 2/20 0.37
F11 P03951 1/20 0.36
TRPV1 Q8NER1 3/20 0.35
MGLL Q99685 1/20 0.35
ENPP2 Q13822 2/20 0.33
CXCR1 P25024 1/20 0.32
CXCR2 P25025 1/20 0.32
CSK P41240 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3865771 0.83 ENPP2 (0.44) LPLLIPGMGLLENPP2CXCR1
SCHEMBL5662615 0.80 LOXL2 (0.35) KDM4ECA2CA1
SCHEMBL643420 0.80 MAPT (0.38)
SCHEMBL5780510 0.80 ALDH1A1 (0.38)
SCHEMBL7763429 0.79 MEN1 (0.41)
SCHEMBL11503093 0.79 RXRA (0.41) KDM4ECA2
SCHEMBL5603701 0.79 ALDH1A1 (0.43)
SCHEMBL6376616 0.78 PPARA (0.44) CA2
SCHEMBL403826 0.77 TAAR1 (0.47)
SCHEMBL6370660 0.77 MEN1 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020207352-A1 TRIAZINE BENZIMIDAZOLE COMPOUNDS AND MEDICAL USE THEREOF 四川科伦博泰生物医药股份有限公司 2020-10-15 WO disclosed
EP-1924561-B1 6-ARYLALKYLAMINO- 2,3,4,5-TETRAHYDRO-1H-BENZO[D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS LILLY CO ELI (US) 2012-11-14 EP disclosed