Methylthiouracil

Methylthiouracil

SCHEMBL13723723

CCCSn1ccc(=O)[nH]c1=O.Cc1cc(=O)[nH]c(=S)[nH]1

nearest known ligand 0.50

Full drug profile on Sugi Atlas →

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.50
LPO P22079 2/20 0.50
PTGS1 P23219 1/20 0.50
KMT2A Q03164 1/20 0.39
MPO P05164 1/20 0.38
TPO P07202 1/20 0.38
TSHR P16473 1/20 0.38
CYP2C19 P33261 1/20 0.38
TAS2R38 P59533 1/20 0.38
CRBN Q96SW2 2/20 0.33
PKM P14618 1/20 0.32
MAPT P10636 1/20 0.32
LMNA P02545 1/20 0.32
GAA P10253 1/20 0.32
CA1 P00915 1/20 0.32
ALDH1A1 P00352 2/20 0.32
CYB5R3 P00387 1/20 0.32
CYP3A4 P08684 1/20 0.32
DUT P33316 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Propylthiouracil SCHEMBL5493721 0.85 LPO (0.59) SMN1; SMN2LPOPTGS1KMT2AMPO
SCHEMBL954608 0.84 CRBN (0.46) CRBNPKMDUT
Thiourea SCHEMBL29139741 0.79 CRBN (0.39) CRBNPKMMAPTLMNAGAA
SCHEMBL4347792 0.74 CRBN (0.47) CRBNPKMLMNAALDH1A1DUT
SCHEMBL16671886 0.74 GPR84 (0.43) SMN1; SMN2CYP2C19CRBNPKM
SCHEMBL8653846 0.73 GPR84 (0.46) CYP2C19CRBNPKM
SCHEMBL8656959 0.71 CRBN (0.48) CRBNPKMLMNAALDH1A1DUT
Methylthiouracil SCHEMBL159989 0.71
Methimazole SCHEMBL8813156 0.69 CRBN (0.39) CRBNPKMDUT
Methylthiouracil SCHEMBL5798462 0.69 SMN1; SMN2 (0.95) SMN1; SMN2LPOPTGS1KMT2AMPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2699572-A1 HETEROCYCLIC COMPOUNDS AS KINASE INHIBITORS Origenis GmbH (DE) 2014-02-26 EP disclosed
EP-2699579-A1 PYRAZOLO [4, 3-D]PYRIMIDINES USEFUL AS KINASE INHIBITORS Origenis GmbH (DE) 2014-02-26 EP disclosed
WO-2012143143-A1 HETEROCYCLIC COMPOUNDS AS KINASE INHIBITORS ORIGENIS GMBH (DE) 2012-10-26 WO disclosed
WO-2012143144-A1 PYRAZOLO [4, 3-D] PYRIMIDINES USEFUL AS KINASE INHIBITORS ORIGENIS GMBH (DE) 2012-10-26 WO disclosed