SCHEMBL13735009

SCHEMBL13735009

CN1CCC(c2ccnn2-c2ccc(N3CCOCC3)cc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
MAPT P10636 5/20 0.40
HTT P42858 4/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
KDM4E B2RXH2 3/20 0.40
HSD17B10 Q99714 2/20 0.40
TP53 P04637 2/20 0.40
MAPK1 P28482 2/20 0.40
USP2 O75604 1/20 0.40
ALOX15 P16050 1/20 0.40
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
NPC1 O15118 1/20 0.37
CYP1A2 P05177 1/20 0.37
RAB9A P51151 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13735207 0.92 GAA (0.44) ALDH1A1SMN1; SMN2MAPTMEN1KMT2A
SCHEMBL13734645 0.90 CHKA (0.39) ALDH1A1SMN1; SMN2MAPTMEN1KMT2A
SCHEMBL13735126 0.83 DRD4 (0.43) SMN1; SMN2NPC1RAB9AGAAMAPK11
SCHEMBL8038871 0.77 QDPR (0.47) ALDH1A1SMN1; SMN2MAPTHTTMEN1
SCHEMBL13733633 0.75 QDPR (0.42) LMNA
SCHEMBL13734830 0.74 NT5E (0.45)
SCHEMBL17001804 0.72 GAA (0.46) SMN1; SMN2HTTKDM4EGAA
SCHEMBL10161185 0.72 GRM2 (0.45) ALDH1A1SMN1; SMN2MAPTHTTMEN1
SCHEMBL13734629 0.71 ROCK2 (0.45)
SCHEMBL14922321 0.71 ALDH1A1 (0.63) ALDH1A1SMN1; SMN2MAPTHTTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2699579-A1 PYRAZOLO [4, 3-D]PYRIMIDINES USEFUL AS KINASE INHIBITORS Origenis GmbH (DE) 2014-02-26 EP claimed
WO-2012143144-A1 PYRAZOLO [4, 3-D] PYRIMIDINES USEFUL AS KINASE INHIBITORS ORIGENIS GMBH (DE) 2012-10-26 WO claimed