SCHEMBL13734830

SCHEMBL13734830

CN1CCC(c2ccnn2-c2ccc3cn[nH]c3c2)CC1

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NT5E P21589 16/20 0.45
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
PDGFRB P09619 2/20 0.38
PDGFRA P16234 2/20 0.38
EGFR P00533 1/20 0.38
FGFR1 P11362 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13734629 0.91 ROCK2 (0.45) SLC6A2SLC6A4SLC6A3
SCHEMBL13735009 0.74 ALDH1A1 (0.40)
SCHEMBL13733633 0.73 QDPR (0.42)
SCHEMBL13735207 0.73 GAA (0.44)
SCHEMBL13735126 0.73 DRD4 (0.43)
SCHEMBL5095062 0.73 FGFR1 (0.56) SLC6A2SLC6A4SLC6A3PDGFRBPDGFRA
SCHEMBL13734645 0.72 CHKA (0.39)
SCHEMBL13734849 0.68 DRD4 (0.47)
SCHEMBL9917339 0.68 SLC6A2 (0.55) SLC6A2SLC6A4SLC6A3
SCHEMBL3537019 0.68 ALDH1A1 (0.71)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2699579-A1 PYRAZOLO [4, 3-D]PYRIMIDINES USEFUL AS KINASE INHIBITORS Origenis GmbH (DE) 2014-02-26 EP disclosed
WO-2012143144-A1 PYRAZOLO [4, 3-D] PYRIMIDINES USEFUL AS KINASE INHIBITORS ORIGENIS GMBH (DE) 2012-10-26 WO disclosed