SCHEMBL13746012

SCHEMBL13746012

Cc1nc([C@H]2CC[C@@H](C(F)(F)F)CC2)c(-c2ccc(C#N)nc2)c(=O)[nH]1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.36
PDE2A O00408 6/20 0.35
DGAT1 O75907 1/20 0.35
KDM5B Q9UGL1 1/20 0.34
PDE9A O76083 1/20 0.33
PI4KB Q9UBF8 1/20 0.33
PDE4A P27815 2/20 0.33
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33
TYK2 P29597 1/20 0.33
JAK3 P52333 1/20 0.33
SYK P43405 1/20 0.33
CXCR2 P25025 1/20 0.32
CCR6 P51684 1/20 0.32
VHL P40337 1/20 0.32
LCAT P04180 1/20 0.32
SPR P35270 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13746898 0.85 HSD11B1 (0.39) PDE2APDE9ACXCR2
SCHEMBL4020404 0.85 PDE2A (0.49) PIK3CAPDE2AKDM5BPDE9API4KB
SCHEMBL13746667 0.85 PDE2A (0.37) PIK3CAPDE2API4KBJAK2JAK1
SCHEMBL4023133 0.81 PDE2A (0.37) PDE2API4KBJAK2JAK1TYK2
SCHEMBL4023129 0.81 PDE2A (0.37) PDE2API4KBJAK2JAK1TYK2
SCHEMBL13747129 0.80 TYMS (0.38) PDE2A
SCHEMBL13746627 0.76 USP1 (0.34) PIK3CAPDE2ASPR
SCHEMBL4753259 0.75 PIK3CA (0.35) PIK3CADGAT1KDM5BPDE9API4KB
SCHEMBL13746091 0.74 DYRK1A (0.35) PDE2APDE4ASPR
SCHEMBL4028394 0.74 BRD4 (0.38) PDE2ASPR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009100403-A1 SUBSTITUTED ARYL PYRIMIDINONES NEUROGEN CORPORATION (US) 2009-08-13 WO disclosed