SCHEMBL13748718

SCHEMBL13748718

O=C(O)c1cc(Cl)c(Cl)cc1C(=O)N1CCc2cc3c(cc2C1c1ccccn1)OCCO3

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 3/20 0.39
HHAT Q5VTY9 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
HTT P42858 1/20 0.37
MAPT P10636 3/20 0.35
NPSR1 Q6W5P4 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
TSHR P16473 3/20 0.35
GRIN2C Q14957 1/20 0.35
POLB P06746 1/20 0.34
PDE5A O76074 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
NPC1 O15118 1/20 0.34
PKM P14618 1/20 0.34
RAB9A P51151 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13809015 0.94 KIF11 (0.45) KIF11HHATHTTMAPTNPSR1
SCHEMBL13809014 0.85 KIF11 (0.48) KIF11HHATMAPTNPSR1L3MBTL1
SCHEMBL13809017 0.82 KIF11 (0.50) KIF11HHATMEN1KMT2AMAPT
SCHEMBL13809005 0.77 KIF11 (0.50) KIF11KMT2AHTTTSHRGRIN2C
SCHEMBL13809025 0.76 KIF11 (0.42) KIF11MEN1KMT2AGRIN2CSMN1; SMN2
SCHEMBL13748440 0.73 MAPT (0.66) MAPTNPSR1L3MBTL1POLBPKM
SCHEMBL11713375 0.69 TRPV1 (0.51) KIF11MEN1KMT2AHTTMAPT
SCHEMBL13809243 0.69 KIF11 (0.53) KIF11MEN1KMT2AGRIN2CALDH1A1
SCHEMBL10025906 0.64 OPRD1 (0.39) HTTNPSR1TSHRGRIN2CPOLB
SCHEMBL11718509 0.63 KIF11 (0.59) KIF11HTTMAPTNPSR1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009102377-A2 ANTIBIOTIC TETRAHYDRO-BETA-CARBOLINE DERIVATIVES MAXTHERA INC. (US) 2009-08-20 WO disclosed
WO-2009073545-A2 TETRAHYDRO-ISOQUINOLINE PPAT INHIBITORS AS ANTIBACTERIAL AGENTS MAXTHERA, INC. (US) 2009-06-11 WO disclosed