SCHEMBL13748940

SCHEMBL13748940

CBc1cnc2c(c1)OCC(=O)N2

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MMP12 P39900 1/20 0.39
PARP1 P09874 1/20 0.36
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
NSD2 O96028 1/20 0.34
GAA P10253 1/20 0.34
ALDH1A1 P00352 3/20 0.33
MAPT P10636 3/20 0.33
NR3C2 P08235 2/20 0.33
LMNA P02545 2/20 0.33
KCNQ1 P51787 1/20 0.33
KCNH2 Q12809 1/20 0.33
CACNA1C Q13936 1/20 0.33
RAB9A P51151 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10283759 0.80 MMP12 (0.49) MMP12PARP1CYP11B1CYP11B2ALDH1A1
SCHEMBL859012 0.76 MMP12 (0.38) MMP12PARP1CYP11B1CYP11B2GAA
SCHEMBL3082129 0.76 ALDH1A1 (0.38) MMP12PARP1CYP11B1CYP11B2ALDH1A1
SCHEMBL18307151 0.76 MMP12 (0.38) MMP12PARP1CYP11B1CYP11B2GAA
SCHEMBL7958200 0.76 MMP12 (0.38) MMP12PARP1CYP11B1CYP11B2GAA
SCHEMBL15979057 0.76 NR3C2 (0.39) MMP12CYP11B1CYP11B2NR3C2KCNH2
SCHEMBL7326455 0.76 PARP1 (0.39) MMP12PARP1CYP11B1CYP11B2NSD2
SCHEMBL19430275 0.76 MMP12 (0.39) MMP12PARP1CYP11B1CYP11B2NSD2
SCHEMBL14804046 0.76 MMP12 (0.39) MMP12PARP1CYP11B1CYP11B2ALDH1A1
SCHEMBL13662161 0.76 PARP1 (0.52) MMP12PARP1CYP11B1CYP11B2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009100536-A1 INHIBITORS OF KINASE ACTIVITY WITH 1,2-DI-CYCLYL SUBSTITUTED ALKYNE STRUCTURES METHYLGENE INC. (CA) 2009-08-20 WO disclosed