SCHEMBL7326455

SCHEMBL7326455

C[Sn](C)(C)c1cnc2c(c1)OCC(=O)N2

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.39
MMP12 P39900 1/20 0.39
CYP11B1 P15538 2/20 0.35
CYP11B2 P19099 2/20 0.35
NR3C2 P08235 5/20 0.33
MAPT P10636 3/20 0.33
ALDH1A1 P00352 3/20 0.33
LMNA P02545 1/20 0.33
RXFP1 Q9HBX9 1/20 0.32
NSD2 O96028 1/20 0.32
PDE3B Q13370 3/20 0.32
PDE3A Q14432 3/20 0.32
PKM P14618 1/20 0.32
KMT2A Q03164 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10283759 0.80 MMP12 (0.49) PARP1MMP12CYP11B1CYP11B2NR3C2
SCHEMBL13662161 0.79 PARP1 (0.52) PARP1MMP12CYP11B1CYP11B2NR3C2
SCHEMBL3082129 0.76 ALDH1A1 (0.38) PARP1MMP12CYP11B1CYP11B2NR3C2
SCHEMBL859012 0.76 MMP12 (0.38) PARP1MMP12CYP11B1CYP11B2NR3C2
SCHEMBL15979057 0.76 NR3C2 (0.39) MMP12CYP11B1CYP11B2NR3C2
SCHEMBL7958200 0.76 MMP12 (0.38) PARP1MMP12CYP11B1CYP11B2NR3C2
SCHEMBL18307151 0.76 MMP12 (0.38) PARP1MMP12CYP11B1CYP11B2NR3C2
SCHEMBL13748940 0.76 MMP12 (0.39) PARP1MMP12CYP11B1CYP11B2NR3C2
SCHEMBL19430275 0.76 MMP12 (0.39) PARP1MMP12CYP11B1CYP11B2NR3C2
SCHEMBL14804046 0.76 MMP12 (0.39) PARP1MMP12CYP11B1CYP11B2NR3C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4906629-A Pyridazinone and pyrazolone compounds, cardiotonic compositions including same, and their uses RORER PHARMACEUTICAL CORPORATION (US) 1990-03-06 US disclosed
US-4829066-A CONGESTIVE HEART FAILURE RORER PHARMACEUTICAL CORPORATION (US) 1989-05-09 US disclosed
WO-1988008706-A1 PYRIDOOXAZINONE-PYRIDAZINONE AND PYRAZOLONE COMPOUNDS, CARDIOTONIC COMPOSITIONS INCLUDING THE SAME, AND THEIR USE RORER INTERNATIONAL (OVERSEAS) INC. (US) 1988-11-17 WO disclosed