SCHEMBL1375014

SCHEMBL1375014

OCc1cccnc1Nc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 4/20 0.56
KMT2A Q03164 6/20 0.51
MEN1 O00255 5/20 0.51
MAPT P10636 4/20 0.51
ALDH1A1 P00352 3/20 0.51
GAA P10253 2/20 0.51
ABCG2 Q9UNQ0 3/20 0.45
GRM4 Q14833 1/20 0.45
RAB9A P51151 4/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
CLK1 P49759 1/20 0.42
KDM4E B2RXH2 3/20 0.42
HTT P42858 3/20 0.42
LMNA P02545 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
NPC1 O15118 2/20 0.42
DAPK3 O43293 1/20 0.42
MAP4K4 O95819 1/20 0.42
ABL1 P00519 1/20 0.42
EGFR P00533 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9402422 0.85 RAB9A (0.57) DHODHKMT2AMEN1MAPTALDH1A1
SCHEMBL9402356 0.85 DHODH (0.57) DHODHKMT2AMAPTALDH1A1ABCG2
SCHEMBL1908379 0.82 DHODH (0.56) DHODHKMT2AMEN1MAPTALDH1A1
SCHEMBL5252795 0.82 DHODH (0.51) DHODHKMT2AMEN1MAPTALDH1A1
SCHEMBL9470451 0.82 DHODH (0.51) DHODHKMT2AMEN1MAPTALDH1A1
SCHEMBL9402425 0.81 RAB9A (0.60) KMT2AMEN1MAPTALDH1A1GAA
SCHEMBL9469965 0.81 DHODH (0.48) DHODHKMT2AMEN1MAPTALDH1A1
SCHEMBL10681378 0.81 ABCG2 (0.50) DHODHALDH1A1ABCG2RAB9ASMN1; SMN2
SCHEMBL9402412 0.81 GRM4 (0.52) KMT2AMAPTALDH1A1ABCG2GRM4
SCHEMBL10672819 0.81 LMNA (0.59) KMT2AMEN1MAPTALDH1A1ABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107573340-B Preparation and application of 2-carbamoyl-4-aryl hetero pyridine compound 江西科技师范大学 2020-11-24 CN disclosed
CN-108314682-A The preparation and application of the miscellaneous quinolines of the disubstituted -4- virtues of 6,7- 江西科技师范大学 2018-07-24 CN disclosed
EP-2394995-B1 RING-FUSED 2-PYRIDONE DERIVATIVES AND HERBICIDES KUMIAI CHEMICAL INDUSTRY CO (JP) 2014-01-15 EP disclosed
US-8334236-B2 Ring-fused 2-pyridone derivatives and herbicides KUMIAI CHEMICAL INDUSTRY CO., LTD. (JP) 2012-12-18 US disclosed
EP-2394995-A1 RING-FUSED 2-PYRIDONE DERIVATIVES AND HERBICIDES Kumiai Chemical Industry CO., LTD. (JP) 2011-12-14 EP disclosed
US-20110287937-A1 RING-FUSED 2-PYRIDONE DERIVATIVES AND HERBICIDES IHARA CHEMICAL INDUSTRY CO., LTD. (JP) 2011-11-24 US disclosed
US-5519037-A N-cyanoamidine derivatives as anti-influenza agents AMERICAN HOME PRODUCTS CORPORATION (US) 1996-05-21 US disclosed
US-5475012-A Antiviral against influenza A AMERICAN HOME PRODUCTS CORPORATION (US) 1995-12-12 US disclosed
US-5380734-A N-cyanoamidine derivatives as anti-influenza agents AMERICAN HOME PRODUCTS CORPORATION (US) 1995-01-10 US disclosed
US-5364860-A Naphthyridine compounds which inhibit tyrosine kinase and their pharmaceutical compositions LABORATOIRES UPSA (FR) 1994-11-15 US disclosed
WO-1991018902-A1 SUBSTITUTED 1-H-PYRROLO[2,3-b]PYRIDINE-3-CARBOXAMIDES SCHERING CORPORATION (US) 1991-12-12 WO disclosed
US-5023265-A Antiinflammatory agent; inhibits both 5-lipoxygenase and cyclooxygenase; rheumatoid arthritis, bursitis, tendonitis, gout; side effect reduction SCHERING CORPORATION (US) 1991-06-11 US disclosed
US-4009166-A ANTIINFLAMMATORY AGENTS, ANALGESICS, CNS DEPRESSANTS HISAMITSU PHARMACEUTICAL CO., INC. (JA) 1977-02-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110287937-A1 RING-FUSED 2-PYRIDONE DERIVATIVES AND HERBICIDES CBR3, CBR1, CHRM1 DHODH 780/4885KMT2A 2625/4885MEN1 4177/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.