SCHEMBL1375494

SCHEMBL1375494

CCOC(=O)c1cc2cccnc2n(-c2ccccc2)c1=O

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MET P08581 3/20 0.52
ALDH1A1 P00352 4/20 0.52
KDM4E B2RXH2 2/20 0.52
HSD17B10 Q99714 1/20 0.52
MAPT P10636 2/20 0.51
CSF1R P07333 1/20 0.48
GAA P10253 2/20 0.48
TP53 P04637 1/20 0.47
ELANE P08246 1/20 0.47
ALOX15 P16050 1/20 0.46
PNP P00491 1/20 0.46
HTT P42858 1/20 0.46
HPGD P15428 2/20 0.45
POLB P06746 1/20 0.45
GLA P06280 1/20 0.45
ADORA2A P29274 1/20 0.45
ADORA1 P30542 1/20 0.45
RECQL P46063 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3517555 0.84 ELANE (0.49) ALDH1A1KDM4EGAAELANEHTT
SCHEMBL1372818 0.84 AHR (0.55) ALDH1A1KDM4EHSD17B10GAAELANE
SCHEMBL1376319 0.84 ELANE (0.44) METALDH1A1KDM4EHSD17B10MAPT
SCHEMBL1374001 0.83 CNR1 (0.59) ALDH1A1KDM4EHSD17B10GAAHPGD
SCHEMBL15334959 0.82 CNR2 (0.49) ALDH1A1KDM4EMAPTGAAELANE
SCHEMBL1375442 0.82 ALDH1A1 (0.48) ALDH1A1KDM4EHSD17B10MAPTGAA
SCHEMBL1375742 0.82 MET (0.52) METALDH1A1
SCHEMBL1376548 0.81 ELANE (0.43) ALDH1A1KDM4EHSD17B10MAPTGAA
SCHEMBL17603562 0.81 MAOB (0.48) ALDH1A1KDM4EMAPTGAAELANE
Hydrochloric Acid SCHEMBL1373870 0.81 MET (0.51) METALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107573340-B Preparation and application of 2-carbamoyl-4-aryl hetero pyridine compound 江西科技师范大学 2020-11-24 CN disclosed
EP-3067356-B1 PYRROLO PYRIMIDINE DERIVATIVE ONO PHARMACEUTICAL CO (JP) 2018-07-04 EP disclosed
US-9586967-B2 Pyrrolo pyrimidine derivative ONO PHARMACEUTICAL CO., LTD. (JP) 2017-03-07 US disclosed
US-20160264579-A1 PYRROLO PYRIMIDINE DERIVATIVE ONO PHARMACEUTICAL CO., LTD. (JP) 2016-09-15 US disclosed
EP-3067356-A1 PYRROLO PYRIMIDINE DERIVATIVE ONO Pharmaceutical Co., Ltd. (JP) 2016-09-14 EP disclosed
EP-2394995-B1 RING-FUSED 2-PYRIDONE DERIVATIVES AND HERBICIDES KUMIAI CHEMICAL INDUSTRY CO (JP) 2014-01-15 EP disclosed
US-8334236-B2 Ring-fused 2-pyridone derivatives and herbicides KUMIAI CHEMICAL INDUSTRY CO., LTD. (JP) 2012-12-18 US disclosed
EP-2394995-A1 RING-FUSED 2-PYRIDONE DERIVATIVES AND HERBICIDES Kumiai Chemical Industry CO., LTD. (JP) 2011-12-14 EP disclosed
US-20110287937-A1 RING-FUSED 2-PYRIDONE DERIVATIVES AND HERBICIDES IHARA CHEMICAL INDUSTRY CO., LTD. (JP) 2011-11-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160264579-A1 PYRROLO PYRIMIDINE DERIVATIVE AXL, FLT3, TYRO3 MET 398/4885ALDH1A1 3360/4885KDM4E 1727/4885
US-20110287937-A1 RING-FUSED 2-PYRIDONE DERIVATIVES AND HERBICIDES CBR3, CBR1, CHRM1 MET 1467/4885ALDH1A1 623/4885KDM4E 2575/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.