SCHEMBL13765784

SCHEMBL13765784

CC(C)(C)c1cncc(NC(=O)C2CC2)n1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ATAD2 Q6PL18 1/20 0.50
HPGD P15428 1/20 0.47
ADORA2B P29275 3/20 0.46
CYP3A4 P08684 2/20 0.46
ADORA2A P29274 2/20 0.46
CYP2D6 P10635 1/20 0.46
ABL1 P00519 10/20 0.44
RAB9A P51151 1/20 0.42
RXFP1 Q9HBX9 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
GLA P06280 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14642749 0.85 ADORA2B (0.45) ATAD2HPGDADORA2BCYP3A4ADORA2A
SCHEMBL13765787 0.80 KDM4E (0.44) ADORA2BRAB9AL3MBTL1CYP1A2
SCHEMBL16938290 0.79 HPGD (0.51) HPGDADORA2BCYP3A4ADORA2ACYP2D6
SCHEMBL10068141 0.78 HPGD (0.70) ATAD2HPGDADORA2BADORA2AABL1
SCHEMBL13765794 0.78 ALDH1A1 (0.46) ABL1RAB9A
SCHEMBL23089548 0.76 HPGD (0.51) HPGDADORA2BCYP3A4ADORA2ACYP2D6
SCHEMBL22529508 0.76 HPGD (0.51) HPGDADORA2BCYP3A4ADORA2ACYP2D6
SCHEMBL17194984 0.74 ATAD2 (0.49) ATAD2HPGDADORA2AABL1RAB9A
SCHEMBL77715 0.72 ATAD2 (0.89) ATAD2HPGDRAB9A
SCHEMBL15274645 0.72 ABL1 (0.47) ATAD2HPGDABL1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8461167-B2 Acetylenic heteroaryl compounds ARIAD PHARMACEUTICALS, INC. (US) 2013-06-11 US disclosed
US-20090176781-A1 Acetylenic Heteroaryl Compounds ARIAD PHARMACEUTICALS, INC. 2009-07-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090176781-A1 Acetylenic Heteroaryl Compounds NAT1, AADAC, ACACA ATAD2 1370/4885HPGD 551/4885ADORA2B 1263/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.