SCHEMBL1376732

SCHEMBL1376732

N#Cc1cccc(C(CNCCNC(=O)O)(c2cccnc2)c2cccnc2)c1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 5/20 0.39
NAMPT P43490 2/20 0.38
BRAF P15056 1/20 0.38
GRM5 P41594 5/20 0.37
CYP3A4 P08684 2/20 0.37
CYP3A5 P20815 2/20 0.37
SGMS2 Q8NHU3 1/20 0.37
SLC22A12 Q96S37 1/20 0.36
KCNA5 P22460 2/20 0.36
ATR Q13535 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1377411 0.75 DGAT2 (0.56) NAMPT
SCHEMBL1381950 0.72 CYP1A2 (0.42) VNN1GRM5CYP3A4
SCHEMBL4198056 0.72 CYP3A4 (0.36) VNN1NAMPTBRAFGRM5CYP3A4
SCHEMBL1376729 0.70 KCNA5 (0.46) VNN1NAMPTBRAFGRM5SGMS2
SCHEMBL1378017 0.69 GRM5 (0.43) VNN1BRAFGRM5ATR
SCHEMBL3819011 0.65 HSD11B1 (0.39) NAMPTGRM5CYP3A4SLC22A12KCNA5
SCHEMBL4184873 0.65 CYP3A4 (0.44) VNN1CYP3A4CYP3A5SGMS2KCNA5
SCHEMBL2007111 0.65 CNR1 (0.62) VNN1
SCHEMBL1246685 0.62 SCN9A (0.52)
SCHEMBL17237438 0.62 NPC1 (0.67) VNN1NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4719745-B2 2011-07-06 JP claimed
EP-1781635-A4 POTASSIUM CHANNEL INHIBITORS MERCK & CO INC (US) 2009-02-25 EP claimed
EP-1781635-A2 POTASSIUM CHANNEL INHIBITORS Merck & Co., Inc. (US) 2007-05-09 EP claimed
WO-2006015159-A2 POTASSIUM CHANNEL INHIBITORS MERCK & CO., INC. (US) 2006-02-09 WO claimed