SCHEMBL13769798

SCHEMBL13769798

CCOC(=O)[C@@H]1CCCN(c2ccc(-c3nc(N)c(C)nc3C)cc2)C1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SHMT2 P34897 1/20 0.49
ALDH1A1 P00352 7/20 0.48
KDM4E B2RXH2 6/20 0.47
MAPT P10636 6/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
HPGD P15428 2/20 0.47
TP53 P04637 2/20 0.47
HSD17B10 Q99714 2/20 0.47
HTT P42858 1/20 0.47
MCL1 Q07820 1/20 0.47
GAA P10253 1/20 0.46
F10 P00742 2/20 0.46
ATM Q13315 1/20 0.45
NPSR1 Q6W5P4 3/20 0.45
MAPK1 P28482 2/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
POLB P06746 1/20 0.45
NPC1 O15118 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13769799 1.00 SHMT2 (0.49) SHMT2ALDH1A1KDM4EMAPTSMN1; SMN2
SCHEMBL13769245 0.88 LGMN (0.56) SHMT2ALDH1A1KDM4EMAPTTP53
SCHEMBL5538159 0.85 KDM4E (0.58) SHMT2ALDH1A1KDM4EMAPTSMN1; SMN2
SCHEMBL5532095 0.85 KDM4E (0.58) SHMT2ALDH1A1KDM4EMAPTSMN1; SMN2
SCHEMBL21848213 0.81 SHMT2 (0.59) SHMT2ALDH1A1KDM4ESMN1; SMN2L3MBTL1
SCHEMBL29891157 0.78 ALDH1A1 (0.54) SHMT2ALDH1A1KDM4EMAPTSMN1; SMN2
SCHEMBL22149667 0.78 ALDH1A1 (0.54) SHMT2ALDH1A1KDM4EMAPTSMN1; SMN2
SCHEMBL16880167 0.78 ALDH1A1 (0.54) SHMT2ALDH1A1KDM4EMAPTSMN1; SMN2
SCHEMBL4684573 0.77 ALDH1A1 (0.58) SHMT2ALDH1A1KDM4EMAPTSMN1; SMN2
SCHEMBL31175186 0.77 ALDH1A1 (0.70) ALDH1A1KDM4ESMN1; SMN2L3MBTL1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081195-A1 CARBAMOYL COMPOUNDS AS DGAT1 INHIBITORS 190 ASTRAZENECA AB (SE) 2009-07-02 WO disclosed