SCHEMBL1378463

SCHEMBL1378463

Nc1ccnc(CC(c2cccnc2)(c2cccnc2)c2cccc(Cl)c2)n1

nearest known ligand 0.48

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 4/20 0.48
RORC P51449 13/20 0.40
KCNA5 P22460 1/20 0.37
SCN5A Q14524 1/20 0.37
SCN9A Q15858 1/20 0.37
KIF11 P52732 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3813461 0.83 CYP19A1 (0.45) CYP19A1RORC
SCHEMBL1377766 0.68 CYP19A1 (0.49) CYP19A1KCNA5
SCHEMBL3819616 0.68 KMO (0.39) CYP19A1KCNA5KIF11
SCHEMBL4191094 0.68 CYP19A1 (0.52) CYP19A1RORCKIF11
SCHEMBL1381592 0.67 CYP19A1 (0.41) CYP19A1
SCHEMBL6000000 0.67 CYP19A1 (0.62) CYP19A1RORC
SCHEMBL5999722 0.66 CYP19A1 (0.57) CYP19A1RORC
SCHEMBL1380492 0.66 KIF11 (0.35) CYP19A1KIF11
SCHEMBL1380977 0.65 CYP3A4 (0.41) CYP19A1
SCHEMBL4194326 0.65 CYP19A1 (0.49) CYP19A1KCNA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4719744-B2 2011-07-06 JP claimed
EP-1776355-A4 POTASSIUM CHANNEL INHIBITORS MERCK & CO INC (US) 2009-08-12 EP claimed
EP-1776355-A2 POTASSIUM CHANNEL INHIBITORS Merck & Co., Inc. (US) 2007-04-25 EP claimed
WO-2006014877-A2 POTASSIUM CHANNEL INHIBITORS MERCK & CO., INC. (US) 2006-02-09 WO claimed