SCHEMBL1380488

SCHEMBL1380488

O=C(O)Cc1c[nH]c2cc(NCCCC#Cc3ccc(OC(F)(F)F)cc3)ccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GOT1 P17174 1/20 0.43
CDK2 P24941 2/20 0.41
KDM4E B2RXH2 1/20 0.41
TRPV1 Q8NER1 5/20 0.40
MAPT P10636 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38
STING1 Q86WV6 1/20 0.37
MMP2 P08253 1/20 0.36
MMP9 P14780 1/20 0.36
TSHR P16473 2/20 0.36
LMNA P02545 2/20 0.36
PTBP1 P26599 1/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.35
HTR6 P50406 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1378534 0.88 PPARD (0.41) GOT1CDK2KDM4ETRPV1MTNR1A
SCHEMBL1379245 0.81 KDM4E (0.50) KDM4ETRPV1MTNR1AMTNR1BTSHR
SCHEMBL1378359 0.79 PPARD (0.43) CDK2KDM4ETSHR
SCHEMBL1383911 0.79 KDM4E (0.41) GOT1CDK2KDM4ETRPV1MTNR1A
SCHEMBL1379036 0.79 KDM4E (0.41) GOT1CDK2KDM4ETRPV1MEN1
SCHEMBL1377718 0.78 KDM4E (0.39) GOT1CDK2KDM4ETRPV1MMP2
SCHEMBL5177050 0.77 PKM (0.44) GOT1TRPV1MAPTMEN1KMT2A
SCHEMBL5176046 0.76 PKM (0.42) GOT1TRPV1MAPTMEN1KMT2A
SCHEMBL5177928 0.76 KDM4E (0.39) GOT1CDK2KDM4ETRPV1TSHR
SCHEMBL5177101 0.74 PPARD (0.36) GOT1CDK2KDM4ETRPV1PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4629106-B2 2011-02-09 JP claimed
JP-2008509947-A 2008-04-03 JP claimed
EP-1781608-A1 INDOLE DERIVATIVES COMPRISING AN ACETYLENE GROUP AS PPAR ACTIVATORS F.HOFFMANN-LA ROCHE AG (CH) 2007-05-09 EP claimed
WO-2006018174-A1 INDOLE DERIVATIVES COMPRISING AN ACETYLENE GROUP AS PPAR ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2006-02-23 WO claimed