SCHEMBL5176046

SCHEMBL5176046

CCOC(=O)Cc1c[nH]c2cc(NC(=O)CCC#Cc3ccc(OC(F)(F)F)cc3)ccc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.42
POLB P06746 1/20 0.41
MAPT P10636 5/20 0.41
ALDH1A1 P00352 4/20 0.40
LMNA P02545 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
GOT1 P17174 1/20 0.40
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
GSK3B P49841 1/20 0.38
TP53 P04637 1/20 0.37
XBP1 P17861 1/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2C19 P33261 2/20 0.36
MCHR1 Q99705 2/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
TSHR P16473 1/20 0.35
STING1 Q86WV6 1/20 0.35
TRPV1 Q8NER1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5177050 0.83 PKM (0.44) PKMPOLBMAPTALDH1A1LMNA
SCHEMBL5176798 0.82 PKM (0.43) PKMPOLBMAPTLMNAGOT1
SCHEMBL9662589 0.78 PKM (0.60) PKMPOLBMAPTALDH1A1LMNA
SCHEMBL5176799 0.78 PKM (0.44) PKMMAPTALDH1A1LMNASMN1; SMN2
SCHEMBL5175332 0.78 PKM (0.42) PKMPOLBMAPTALDH1A1LMNA
SCHEMBL1380488 0.76 GOT1 (0.43) MAPTALDH1A1LMNASMN1; SMN2GOT1
SCHEMBL5177379 0.76 PKM (0.44) PKMMAPTALDH1A1LMNASMN1; SMN2
SCHEMBL5176038 0.75 PKM (0.44) PKMMAPTALDH1A1LMNASMN1; SMN2
SCHEMBL3872201 0.75 LMNA (0.43) POLBMAPTALDH1A1LMNASMN1; SMN2
SCHEMBL1377718 0.74 KDM4E (0.39) ALDH1A1LMNAGOT1CYP2C9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781608-A1 INDOLE DERIVATIVES COMPRISING AN ACETYLENE GROUP AS PPAR ACTIVATORS F.HOFFMANN-LA ROCHE AG (CH) 2007-05-09 EP disclosed
WO-2006018174-A1 INDOLE DERIVATIVES COMPRISING AN ACETYLENE GROUP AS PPAR ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2006-02-23 WO disclosed