SCHEMBL13808741

SCHEMBL13808741

COc1ccc(OC)c2c1CCN(Cc1cccc(-c3nnn[nH]3)c1)C2c1cccc(Cl)c1Cl

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
RORC P51449 2/20 0.35
CNR2 P34972 3/20 0.35
CNR1 P21554 2/20 0.35
HCRTR1 O43613 10/20 0.33
HCRTR2 O43614 10/20 0.33
DRD2 P14416 1/20 0.33
DRD4 P21917 1/20 0.33
DRD3 P35462 1/20 0.33
HTR7 P34969 1/20 0.32
LMNA P02545 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13808739 0.93 RORC (0.33) RORCHCRTR1HCRTR2DRD2DRD4
SCHEMBL13809226 0.81 ABCG2 (0.39)
SCHEMBL13808738 0.76 MAPT (0.42) DRD4
SCHEMBL13809231 0.74 GRIN2C (0.39)
SCHEMBL13748958 0.67 TRPM8 (0.57)
SCHEMBL22480510 0.65 MRGPRX4 (0.65)
SCHEMBL2783497 0.65 KDM4E (0.48)
SCHEMBL13809007 0.63 GRIN2C (0.43) LMNA
SCHEMBL2233428 0.63 TSHR (0.34)
SCHEMBL13809244 0.62 GRIN2C (0.36) RORCLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009073545-A2 TETRAHYDRO-ISOQUINOLINE PPAT INHIBITORS AS ANTIBACTERIAL AGENTS MAXTHERA, INC. (US) 2009-06-11 WO disclosed