SCHEMBL13809231

SCHEMBL13809231

COc1ccc(OC)c2c1CCN(C(=O)c1ccccc1-c1nnn[nH]1)C2c1cccc(Cl)c1Cl

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GRIN2C Q14957 1/20 0.39
P2RX7 Q99572 11/20 0.39
PARP1 P09874 1/20 0.36
ABCB1 P08183 1/20 0.34
ABCG2 Q9UNQ0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13809226 0.85 ABCG2 (0.39) GRIN2CP2RX7ABCB1ABCG2
SCHEMBL13809253 0.82 GRIN2C (0.43) GRIN2CP2RX7ABCB1ABCG2
SCHEMBL13809228 0.80 GRIN2C (0.43) GRIN2CP2RX7ABCB1ABCG2
SCHEMBL13809007 0.79 GRIN2C (0.43) GRIN2CP2RX7ABCB1ABCG2
SCHEMBL13809241 0.76 GRIN2C (0.41) GRIN2CP2RX7ABCB1ABCG2
SCHEMBL13808739 0.76 RORC (0.33)
SCHEMBL13808741 0.74 RORC (0.35)
SCHEMBL13809234 0.73 GRIN2C (0.40) GRIN2CABCB1ABCG2
SCHEMBL13809244 0.72 GRIN2C (0.36) GRIN2C
SCHEMBL13809251 0.66 GRIN2C (0.49) GRIN2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009073545-A2 TETRAHYDRO-ISOQUINOLINE PPAT INHIBITORS AS ANTIBACTERIAL AGENTS MAXTHERA, INC. (US) 2009-06-11 WO disclosed