SCHEMBL13809153

SCHEMBL13809153

CCc1nc2c(c(=O)n(C)c(=O)n2C)n1Cc1ccc(F)cc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.69
TSHR P16473 5/20 0.69
HTT P42858 6/20 0.68
LMNA P02545 2/20 0.67
SMN1; SMN2 Q16637 2/20 0.67
MAPK1 P28482 2/20 0.65
GFER P55789 1/20 0.65
HSD17B10 Q99714 4/20 0.64
CASP1 P29466 1/20 0.64
CASP7 P55210 1/20 0.64
ALOX15 P16050 2/20 0.63
USP2 O75604 1/20 0.63
MAPT P10636 4/20 0.62
PCSK9 Q8NBP7 1/20 0.62
NPSR1 Q6W5P4 3/20 0.59
ALDH1A1 P00352 4/20 0.57
KMT2A Q03164 1/20 0.56
POLB P06746 1/20 0.56
HPGD P15428 1/20 0.56
NCOA3 Q9Y6Q9 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13809397 0.86 PCSK9 (0.65) TP53TSHRHTTLMNASMN1; SMN2
SCHEMBL16029366 0.85 HTT (0.61) TP53TSHRHTTLMNASMN1; SMN2
SCHEMBL555962 0.85 HTT (0.74) TP53TSHRHTTLMNASMN1; SMN2
SCHEMBL16079532 0.84 HTT (0.60) TP53TSHRHTTLMNASMN1; SMN2
SCHEMBL7016485 0.82 ALDH1A1 (0.60) TP53TSHRHTTLMNASMN1; SMN2
SCHEMBL17791591 0.79 HSD17B10 (1.00) TP53TSHRHTTLMNASMN1; SMN2
SCHEMBL13939505 0.79 NPSR1 (0.76) TP53TSHRHTTLMNASMN1; SMN2
SCHEMBL13938418 0.78 NPSR1 (0.65) TP53TSHRHTTLMNASMN1; SMN2
SCHEMBL24769080 0.77 PCSK9 (1.00) TP53TSHRHTTLMNASMN1; SMN2
SCHEMBL555168 0.77 DPP4 (0.80) TP53TSHRHTTLMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1319003-B1 XANTHINE PHOSPHODIESTERASE V INHIBITORS SCHERING CORP (US) 2009-06-10 EP disclosed