SCHEMBL7016485

SCHEMBL7016485

CCc1nc2c(c(=O)n(C)c(=O)n2C)n1Cc1ccc(C(=O)c2ccc(Cl)cc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.60
NPSR1 Q6W5P4 4/20 0.60
HTT P42858 3/20 0.60
TSHR P16473 2/20 0.60
RAB9A P51151 1/20 0.60
ATM Q13315 1/20 0.57
MAPT P10636 5/20 0.56
MAPK1 P28482 2/20 0.56
SMN1; SMN2 Q16637 2/20 0.53
HSD17B10 Q99714 2/20 0.52
ALOX15 P16050 1/20 0.52
TP53 P04637 2/20 0.52
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
CASP1 P29466 1/20 0.51
CASP7 P55210 1/20 0.51
MAOA P21397 1/20 0.50
MAOB P27338 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7015626 0.88 HTT (0.67) ALDH1A1NPSR1HTTTSHRRAB9A
SCHEMBL7017271 0.87 TSHR (0.59) ALDH1A1NPSR1HTTTSHRRAB9A
SCHEMBL7016235 0.84 SMN1; SMN2 (0.63) ALDH1A1NPSR1HTTTSHRRAB9A
SCHEMBL8645613 0.83 TSHR (0.47) ALDH1A1NPSR1HTTTSHRRAB9A
SCHEMBL13809153 0.82 TP53 (0.69) ALDH1A1NPSR1HTTTSHRMAPT
SCHEMBL16028537 0.80 TRPC5 (0.63) ALDH1A1NPSR1HTTTSHRRAB9A
SCHEMBL7015623 0.80 TSHR (0.56) ALDH1A1NPSR1HTTTSHRRAB9A
SCHEMBL16029209 0.79 HTT (0.78) ALDH1A1NPSR1HTTTSHRRAB9A
SCHEMBL16029914 0.78 ALDH1A1 (0.60) ALDH1A1NPSR1HTTTSHRRAB9A
SCHEMBL16079534 0.77 ALDH1A1 (0.59) ALDH1A1NPSR1HTTTSHRRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed