SCHEMBL13809228

SCHEMBL13809228

COc1ccc(OC)c2c1CCN(C(=O)c1ccccc1C#N)C2c1cccc(Cl)c1Cl

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRIN2C Q14957 1/20 0.43
ABCG2 Q9UNQ0 3/20 0.38
ABCB1 P08183 1/20 0.38
HTR1D P28221 1/20 0.36
HTR1B P28222 1/20 0.36
P2RX7 Q99572 4/20 0.36
AR P10275 2/20 0.36
HSD11B1 P28845 2/20 0.36
HCRTR1 O43613 1/20 0.35
HCRTR2 O43614 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13809253 0.88 GRIN2C (0.43) GRIN2CABCG2ABCB1HTR1DHTR1B
SCHEMBL13809234 0.85 GRIN2C (0.40) GRIN2CABCG2ABCB1MEN1KMT2A
SCHEMBL13809007 0.84 GRIN2C (0.43) GRIN2CABCG2ABCB1HTR1DHTR1B
SCHEMBL13809241 0.81 GRIN2C (0.41) GRIN2CABCG2ABCB1P2RX7HCRTR1
SCHEMBL13809231 0.80 GRIN2C (0.39) GRIN2CABCG2ABCB1P2RX7
SCHEMBL13809244 0.79 GRIN2C (0.36) GRIN2CMEN1KMT2A
SCHEMBL13808738 0.73 MAPT (0.42)
SCHEMBL13809226 0.72 ABCG2 (0.39) GRIN2CABCG2ABCB1P2RX7HSD11B1
SCHEMBL13809245 0.71 RXFP1 (0.45) GRIN2CMEN1KMT2A
SCHEMBL13809251 0.69 GRIN2C (0.49) GRIN2CMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009073545-A2 TETRAHYDRO-ISOQUINOLINE PPAT INHIBITORS AS ANTIBACTERIAL AGENTS MAXTHERA, INC. (US) 2009-06-11 WO disclosed